The high biological activity of the chromene compounds coupled with the intriguing optical
features of azo chromophores prompted our desire to construct novel derivatives of …

Since the discovery of penicillin, the development and use of antibiotics have promoted safe
and effective control of bacterial infections. However, the number of antibiotic-resistance …

Abstract A series of 5-substituted-1, 3, 4-thiadiazole-based fluoroquinolone derivatives were
designed as potential antibacterial and anticancer agents using a molecular hybridization …

The development of new antimicrobials has always been a research hotspot. In this study, β-
pinene-based derivatives were synthesized, and their antimicrobial activity was evaluated …

With the pressing issue of antibiotic resistance, there is a constant need for new antibiotics.
However, the fact that traditional methods of drug discovery are expensive and time …

In an effort to establish new drug candidates with improved antimicrobial and anticancer
activities, we report here synthesis, molecular modeling, and in vitro biological evaluation of …

Regio‐and stereoselective 1, 3‐dipolar cycloadditions of C‐(chrom‐4‐one‐3‐yl)‐N‐
phenylnitrones (N) with different mono‐substituted, disubstituted, and cyclic dipolarophiles …

Herein, we report the synthesis, characterization, and carbonic anhydrase (CA) inhibition of
the newly synthesized Schiff's bases 4–18 with benzenesulfonamide, methanesulfonamide …

Sustained release dosage forms enable prolonged and continuous release of a drug in the
gastrointestinal tract for medication characterized by a short half lifetime. In this study, the …

Gram‐negative pathogens represent a significant global health threat, while the emergency
and widespread of drug resistance make the situation even worse. As “privileged building …