Recent advances in the synthesis and application of tetrazoles

CS Dai Lingling, GLV Damu, C Zhou - Chinese Journal of Organic …, 2013 - sioc-journal.cn
Tetrazole is an important five-membered aromatic heterocycle with poly-nitrogen electron-
rich planar structural feature. This unique structure endows tetrazole derivatives as drugs …

[HTML][HTML] Цианотиоацетамид–полифункциональный реагент с большими синтетическими возможностями

ВД Дяченко, ИВ Дяченко, ВГ Ненайденко - Успехи химии, 2018 - uspkhim.ru
Аннотация Систематизированы и проанализированы литературные данные по
химическим свойствам α-цианотиоацетамида—удобного исходного реагента для …

Synthesis pharmacological evaluation and docking studies of pyrimidine derivatives

D Giles, K Roopa, FR Sheeba… - European journal of …, 2012 - Elsevier
A new group of pyrimidine derivatives of indane-1, 3-dione were synthesized aiming at the
synthesis of new compounds acting as analgesic, anti-inflammatory and antimicrobial …

Synthesis of 4-aryl-3-methyl-6-oxo-4, 5, 6, 7-tetrahydro-2H-pyrazolo [3, 4-b] pyridine-5-carbonitrile via a one-pot, three-component reaction

A Rahmati - Tetrahedron Letters, 2010 - Elsevier
A one-pot, three-component condensation reaction of an aldehyde, 3-amino-5-
methylpyrazole and ethyl cyanoacetate in ethanol to give 4-aryl-3-methyl-6-oxo-4, 5, 6, 7 …

Design and synthesis of new series of 3‐cyanopyridine and pyrazolopyridine derivatives

RM Keshk - Journal of Heterocyclic Chemistry, 2020 - Wiley Online Library
Abstract Reaction of 3‐cyano‐4, 6‐dimethyl‐2‐pyridone with ethyl chloroacetate afforded
ethyl 2‐([3‐cyano‐4, 6‐dimethylpyridin‐2‐yl] oxy) acetate 2 and ethyl 2‐(3‐cyano‐4, 6 …

[PDF][PDF] 四唑类化合物的合成及应用研究新进展

代玲玲, 崔胜峰, 周成合 - 2013 - researchgate.net
摘要四唑是一种重要的五元芳杂环, 具有多氮富电子的平面结构特征. 这种特殊的结构使得四唑
类化合物作为药物, 炸药, 功能材料等在医学, 农学, 材料科学等众多领域具有广泛的应用前景 …

Synthesis, Antifungal, and Antioxidant Evaluation of New Class of Thiazoloquinazoline Linked by Carbonyl with Nitrile, Phenylacrylonitrile, Pyrazole, Pyrazolo[1,5-a]pyrimidine …

EAM Saleh, SY Kotian, AMAL Dawsari… - Russian Journal of …, 2022 - Springer
A specific route for the synthesis of a novel benzo [4, 5] thiazolo [2, 3-b] quinazoline (IVa–
e),(VIa–e),(VIIa–e),(VIIIa–e),(IXa–e), and (Xa–e) derivatives, where established using …

Synthesis and biological evaluation of 7-trifluoromethylpyrazolo [1, 5-a] pyrimidines as anti-inflammatory and antimicrobial agents

R Aggarwal, E Masan, P Kaushik, D Kaushik… - Journal of Fluorine …, 2014 - Elsevier
A series of 2-H/methyl-3-phenyl-5-alkyl/aryl/heteroaryl-7-trifluoromethylpyrazolo [1, 5-a]
pyrimidines (4a–l) were synthesized by refluxing 3 (5)-amino-4-phenyl-5 (3)-H/methyl-1H …

[HTML][HTML] Synthesis, antiviral activity, and 3D-QSAR study of novel chalcone derivatives containing malonate and pyridine moieties

Z Chen, P Li, D Hu, L Dong, J Pan, L Luo… - Arabian Journal of …, 2019 - Elsevier
Several novel chalcone derivatives containing malonate and pyridine moieties were
synthesized, and their structures were confirmed by 1 H nuclear magnetic resonance, 13 C …

A facile, regioselective synthesis of novel 3-(N-phenylcarboxamide)pyrazolo[1,5-a]pyrimidine analogs in the presence of KHSO in aqueous media assisted by …

S Kaping, I Boiss, LI Singha, P Helissey… - Molecular …, 2016 - Springer
An environmentally benign, simple, efficient, and convenient route is described for the
synthesis of novel pyrazolo [1, 5-a] pyrimidine derivatives under ultrasound irradiation …