As an important branch of the Michael addition reaction, the aza‐Michael addition cascade
reaction has been developed rapidly in recent years. This is because the reaction serves as …

Chiral aza‐heterocycles, as a sort of key frameworks of natural products et al, are deeply
concerned by synthetic chemists. In recent years, catalytic asymmetric reactions of several …

The catalytic enantioselective construction of three-dimensional molecular architectures
from planar aromatics such as quinolines is of great interest and importance from the …

Presented herein is a condition-controlled selective synthesis of pyrazolonyl
spirodihydroquinolines or pyrazolonyl spiroindolines through formal [5+ 1] or [4+ 1] …

An Ir-catalyzed allylic vinylation reaction of allyl carbonates with o-aminostyrene derivatives
has been realized, providing skipped (Z, E)-diene derivatives. With (E)-but-2-ene-1, 4-diyl …

Vinylsulfonium salt chemistry is becoming increasingly attractive in the synthesis of
heterocyclic motifs for its high efficiency and versatility. In this article, we achieved diverse …

Filling a gap in the literature, this book comprehensively reviews catalytic CH addition
reactions of (hetero) aromatic hydrocarbons across carbon-carbon multiple bonds. In so …

A novel one-pot reaction of anilines with acetylenedicarboxylate diesters in the presence of
boron trifluoride, iodine, and trifluoroacetic acid or methylsulfonic acid has been developed …

Determining the activity of a compound and the potential impact on a diseased state is
frequently undertaken using phenotypic or target-based approaches. Phenotypic screens …

Quinolinium ions are engaged in an asymmetric, Ni-catalyzed Suzuki cross-coupling to yield
2-aryl-and 2-heteroaryl-1, 2-dihydroquinolines. Key to the development of this method is the …