Recent progress in the selective fluorinations of some functionalized cycloalkenes

M Nonn, C Paizs, L Kiss - The Chemical Record, 2022 - Wiley Online Library
Organofluorine compounds have had an increasing impact in synthetic organic chemistry
and pharmaceutical research over the past two decades. Their syntheses and the …

Application of 2‐Azabicyclo [2.2. 1] Hept‐5‐En‐3‐One (Vince Lactam) in Synthetic Organic and Medicinal Chemistry

M Nonn, S Fustero, L Kiss - The Chemical Record, 2024 - Wiley Online Library
Azabicyclo [2.2. 1] hept‐5‐en‐3‐one (Vince lactam) is known to be a valuable building block
in synthetic organic chemistry and drug research. It is an important precursor to access of …

Synthesis of New β‐Amino Acid Scaffolds by Means of Ring‐Rearrangement Metathesis

A Semghouli, AM Remete, L Kiss - ChemistrySelect, 2022 - Wiley Online Library
The synthesis of some novel functionalized azaheterocyclic β‐amino esters with multiple
chiral centers via a stereocontrolled synthetic route has been carried out using some …

Application of Metathesis Protocols to the Stereocontrolled Synthesis of some Functionalized β‐Amino Esters and Azaheterocycles

A Semghouli, M Nonn, AM Remete… - The Chemical …, 2023 - Wiley Online Library
In this account our aim was to give an insight into the application of metathesis protocols
(ROM, RCM, RCEYM, CM, RRM) for the synthesis of various azaheterocyclic frameworks …

Extending the substrate scope of palladium-catalyzed arylfluorination of allylic amine derivatives

TT Novák, TCT Nguyen, Á Gömöry… - Journal of Fluorine …, 2024 - Elsevier
Fluorinated molecules often show superior bioactivity or ADME (absorption, distribution,
metabolism, and excretion) properties compared to their non-fluorinated analogues. In fact …

Selective Functionalizations of Cycloalkene‐Fused β‐Lactams and their Transformations into Densely‐Substituted Three‐Dimensional Molecular Entities

M Nonn, L Kiss - Asian Journal of Organic Chemistry, 2023 - Wiley Online Library
Highly‐functionalized, three‐dimensional molecules have had an increasing impact in
synthetic organic chemistry and pharmaceutical research over the past decades. Their …

Attempts on Fluorinative Transformation of Selected Functionalized Cycloalkene Scaffolds through Aziridination/Aziridine-Opening Protocol

TT Novák, Á Gömöry, M Nonn, J Han, L Kiss - Synlett, 2024 - thieme-connect.com
Studies on the transformations of some functionalized cycloalkene derivatives through their
ring olefin-bond aziridination/aziridine opening with fluoride are presented. The selected …

Selective Transformation of 1, 3‐Cyclooctadiene into Novel Functionalized Azaheterocycles, β‐Amino Esters, and Lactams by Means of Ring‐Rearrangement …

A Semghouli, L Drahos, B Volk… - European Journal of …, 2024 - Wiley Online Library
Diversity‐oriented synthesis of some novel functionalized azaheterocyclic β‐amino esters
with multiple chiral centers from 1, 3‐cyclooctadiene‐based β‐amino acids through a …

Extending the Substrate Scope of Palladium-Catalyzed Arylfluorination of Allylic Amine Derivatives

L Kiss, TT Novák, TCT Nguyen, Á Gömöry… - Available at SSRN … - papers.ssrn.com
Fluorinated molecules often show superior bioactivity or ADME (absorption, distribution,
metabolism, and excretion) properties compared to their non-fluorinated analogues. In fact …

[PDF][PDF] Application of metathesis reaction protocols to the stereocontrolled access of some functionalized azaheterocycles

A Semghouli - doktori.bibl.u-szeged.hu
2. Methods The synthesized compounds were separated and purified by column
chromatography on silica gel and by crystallization. The newly prepared compounds were …