[HTML][HTML] Thiazole Ring-The Antimicrobial, Anti-Inflammatory, and Anticancer Active Scaffold

S Hosseininezhad, A Ramazani - Arabian Journal of Chemistry, 2023 - Elsevier
Background Thiazole ring is one of the most important heterocycle scaffolds in organic and
medicinal chemistry due to this scaffold being the backbone of numerous drugs and their …

A retrospect on antimicrobial potential of thiazole scaffold

I Mishra, R Mishra, S Mujwar… - Journal of …, 2020 - Wiley Online Library
Due to its appreciable diversity in biological actions, thiazole and its substituted
components, a significant class of heterocyclic compounds has developed as an influential …

1, 3, 4-thiadiazole scaffold: Anti-microbial agents

T Anthwal, HO Singh, S Nain - Pharmaceutical Chemistry Journal, 2022 - Springer
1, 3, 4-Thiadiazole moiety has various biological activities including anticancer, antidiabetic,
antihypertensive, anti-inflammatory, antiviral, and anti-microbial. Some drugs with …

[PDF][PDF] Antibacterial Activity of Thiazole and its Derivatives: A

P Mohanty, S Behera, R Behura… - … Res. Appl. Chem, 2021 - biointerfaceresearch.com
Thiazoles are one of the most intensively scrutinized classes of 5-membered aromatic
heterocycles. Many natural and synthesized thiazole and its derivatives showed significant …

Diverse biological activities of 1, 3, 4-thiadiazole scaffold

T Anthwal, S Paliwal, S Nain - Chemistry, 2022 - mdpi.com
The chemistry of 1, 3, 4-thiadiazole is one of the most interesting scaffolds for synthesizing
new drug molecules due to their numerous pharmacological activities. Several modifications …

Review on synthetic chemistry and antibacterial importance of thiazole derivatives

A Kashyap, N Adhikari, A Das, A Shakya… - Current drug …, 2018 - ingentaconnect.com
Background: Thiazole is one of the leading heterocyclic five-member ring compounds that
contain nitrogen and sulphur atom. Many natural and/or synthetic compounds contain …

Thiadiazole and Thiazole Derivatives as Potential Antimicrobial Agents

Ц Khamitova, D Berillo, A Lozynskyi… - Mini Reviews in …, 2024 - ingentaconnect.com
Background: This review summarizes data on heterocyclic systems with thiadiazole and
thiazole fragments in molecules as promising antimicrobial agents. Introduction: Thiadiazole …

Thiazole ring—A biologically active scaffold

A Petrou, M Fesatidou, A Geronikaki - Molecules, 2021 - mdpi.com
Background: Thiazole is a good pharmacophore nucleus due to its various pharmaceutical
applications. Its derivatives have a wide range of biological activities such as antioxidant …

Thiazole scaffold: an overview on its synthetic and pharmaceutical aspects

I Mishra, N Sachan - ECS Transactions, 2022 - iopscience.iop.org
Thiazole and its derivatives have risen to prominence as an important scaffold, attracting the
attention of researchers in the area of medicinal chemistry due to their remarkable variety of …

Thiazolotriazoles As Anti-infectives: Design, Synthesis, Biological Evaluation and In Silico Studies

UK Purakkel, G Praveena, VY Madabhushi… - ACS …, 2024 - ACS Publications
The rational design of novel thiazolo [2, 3-c][1, 2, 4] triazole derivatives was carried out
based on previously identified antitubercular hit molecule H127 for discovering potent …