Design and synthesis of oxazepine derivatives from sulfonamide Schiff bases as antimicrobial and antioxidant agents with low cytotoxicity and hemolytic prospective
SA Hassan, DM Aziz, MN Abdullah, AR Bhat… - Journal of Molecular …, 2023 - Elsevier
The eco-friendly sonication and microwave irradiation techniques were used for the straight
forward synthesis of the Schiff base platform from sulfathiazole. Herein, Schiff bases were …
forward synthesis of the Schiff base platform from sulfathiazole. Herein, Schiff bases were …
Synthesis, antibacterial and antioxidant activities of Thiazole-based Schiff base derivatives: a combined experimental and computational study
Abstract Background Thiazole-based Schiff base compounds display significant
pharmacological potential with an ability to modulate the activity of many enzymes involved …
pharmacological potential with an ability to modulate the activity of many enzymes involved …
In vitro and in vivo evaluation of the antimicrobial, antioxidant, cytotoxic, hemolytic activities and in silico POM/DFT/DNA-binding and pharmacokinetic analyses of …
SA Hassan, DM Aziz, MN Abdullah… - Journal of …, 2024 - Taylor & Francis
In this work, Schiff bases and Thiazolidin-4-ones, were synthesized using Sonication and
Microwave techniques, respectively. The Schiff base derivatives (3a–b) were synthesized …
Microwave techniques, respectively. The Schiff base derivatives (3a–b) were synthesized …
Synthesis, antimicrobial and antioxidant evaluation with in silico studies of new thiazole Schiff base derivatives
A series of nineteen thiazole Schiff base derivatives 2a-2s were synthesized (Scheme 1)
and elucidated by spectral analyses (IR, 1 H NMR and HRMS). The evaluation of their …
and elucidated by spectral analyses (IR, 1 H NMR and HRMS). The evaluation of their …
Synthesis, DFT Analysis, and Evaluation of Antibacterial and Antioxidant Activities of Sulfathiazole Derivatives Combined with In Silico Molecular Docking and …
Y Samuel, A Garg, E Mulugeta - Biochemistry Research …, 2021 - Wiley Online Library
Synthetic modifications of sulfathiazole derivatives become an interesting approach to
enhance their biological properties in line with their applications. As a result, sulfathiazole …
enhance their biological properties in line with their applications. As a result, sulfathiazole …
Enhanced synthesis of novel multisubstituted isoxazolidines as potential antimicrobial and antioxidant agents using zinc (II) catalyst, and in silico studies
A Al-Adhreai, M ALSaeedy, A Alrabie… - Journal of Molecular …, 2023 - Elsevier
In the effort of our endeavour to synthesize new heterocyclic bioactive agents, we succeed
the synthesis of a new series of Multisubstituted isoxazolidines (3-(4-substituted)-5-(1H …
the synthesis of a new series of Multisubstituted isoxazolidines (3-(4-substituted)-5-(1H …
Schiff base clubbed benzothiazole: synthesis, potent antimicrobial and MCF-7 anticancer activity, DNA cleavage and computational study
VR Mishra, CW Ghanavatkar, SN Mali… - Journal of …, 2019 - Taylor & Francis
Schiff bases containing benzothiazole unit are synthesized and characterized by 1 H NMR,
13 C NMR, LC–MS, UV–visible and fluorescence spectroscopy methods. Synthesized …
13 C NMR, LC–MS, UV–visible and fluorescence spectroscopy methods. Synthesized …
Synthesis of some novel coumarin isoxazol sulfonamide hybrid compounds, 3D-QSAR studies, and antibacterial evaluation
SN Esfahani, MS Damavandi, P Sadeghi, Z Nazifi… - Scientific reports, 2021 - nature.com
With the progressive and ever-increasing antibacterial resistance pathway, the need for
novel antibiotic design becomes critical. Sulfonamides are one of the more effective …
novel antibiotic design becomes critical. Sulfonamides are one of the more effective …
Design, Synthesis, In Vitro Antimicrobial, Antioxidant Evaluation, and Molecular Docking Study of Novel Benzimidazole and Benzoxazole Derivatives
BB Kashid, AA Ghanwat, VM Khedkar… - Journal of …, 2019 - Wiley Online Library
A series of novel 2‐substituted benzimidazole and benzoxazole derivatives as a potential
antimicrobial and antioxidant agent were synthesized via coupling of N‐methyl‐o …
antimicrobial and antioxidant agent were synthesized via coupling of N‐methyl‐o …
A new series of Schiff bases derived from sulfa drugs and indole-3-carboxaldehyde: Synthesis, characterization, spectral and DFT computational studies
H Ebrahimi, JS Hadi, HS Al-Ansari - Journal of molecular structure, 2013 - Elsevier
A new series of Schiff bases were synthesized for the first time by the condensation of indole-
3-carboxaldehyde with various sulfa drugs including sulfanilamide, sulfapyridine …
3-carboxaldehyde with various sulfa drugs including sulfanilamide, sulfapyridine …