A review on development of bio-active thiosemicarbazide derivatives: Recent advances
There has been substantial attention in the expansion of new thiosemicarbazide derivatives
with diverse biological activities in recent years. Therefore, many scientists have prepared …
with diverse biological activities in recent years. Therefore, many scientists have prepared …
Thiazole derivatives in medicinal chemistry: Recent advancements in synthetic strategies, structure activity relationship and pharmacological outcomes
Thiazole derivatives remains honored heterocycles in the field of medicinal chemistry. This
scaffold has been proven as a universal motif that is present in numerous pharmacologically …
scaffold has been proven as a universal motif that is present in numerous pharmacologically …
Synthesis, characterization, biochemical, and molecular modeling studies of carvacrol‐based new thiosemicarbazide and 1, 3, 4‐thiadiazole derivatives
T Alagöz, FG Çalişkan, HG Bilgiçli… - Archiv der …, 2023 - Wiley Online Library
A series of carvacrol‐based thiosemicarbazide (3a–e) and 1, 3, 4‐thiadiazole‐2‐amine (4a–
e) were designed and synthesized for the first time. The structures were characterized by …
e) were designed and synthesized for the first time. The structures were characterized by …
[HTML][HTML] Exploring the synthesis, structure, spectroscopy and biological activities of novel 4-benzylidene-1-(2-(2, 4-dichloro phenyl) acetyl) thiosemicarbazide …
Background Novel α-amylase inhibitors play a crucial role in managing diabetes and
obesity, contributing to improved public health by addressing these challenging and …
obesity, contributing to improved public health by addressing these challenging and …
Synthetic and medicinal perspective of thiazolidinones: A review
In the modern scenario, thiazolidinone scaffold has emerged as a very potent scaffold as per
its clinical significance concerned. It has attracted the keen interest of the researchers due to …
its clinical significance concerned. It has attracted the keen interest of the researchers due to …
Multifaceted bioactivity of thiosemicarbazide derivatives: Synthesis, characterization, and DFT investigations on inhibition of α-amylase, hydroxyl radical scavenging …
In this study, eight bioactive thiosemicarbazide derivatives (3a-h) were synthesized and
characterized through 1 HNMR, 13 CNMR and Mass spectroscopic techniques. Finally, their …
characterized through 1 HNMR, 13 CNMR and Mass spectroscopic techniques. Finally, their …
Bioactive thiazine and benzothiazine derivatives: green synthesis methods and their medicinal importance
SL Badshah, A Naeem - Molecules, 2016 - mdpi.com
Thiazines are a group of heterocyclic organic compounds that are still largely unexplored for
their pharmacological activities. There are different available methods for the synthesis of …
their pharmacological activities. There are different available methods for the synthesis of …
Synthesis and antiviral properties of novel indole-based thiosemicarbazides and 4-thiazolidinones
G Cihan-Üstündağ, E Gürsoy, L Naesens… - Bioorganic & Medicinal …, 2016 - Elsevier
A novel series of indolylthiosemicarbazides (6a–6g) and their cyclization products, 4-
thiazolidinones (7a–7g), have been designed, synthesized and evaluated, in vitro, for their …
thiazolidinones (7a–7g), have been designed, synthesized and evaluated, in vitro, for their …
A retrospect on antimicrobial potential of thiazole scaffold
Due to its appreciable diversity in biological actions, thiazole and its substituted
components, a significant class of heterocyclic compounds has developed as an influential …
components, a significant class of heterocyclic compounds has developed as an influential …
An overview on synthetic 2-aminothiazole-based compounds associated with four biological activities
M Farouk Elsadek, B Mohamed Ahmed… - Molecules, 2021 - mdpi.com
Amongst sulfur-and nitrogen-containing heterocyclic compounds, the 2-aminothiazole
scaffold is one of the characteristic structures in drug development as this essential …
scaffold is one of the characteristic structures in drug development as this essential …