Cocrystals of pyrazinamide with p-toluenesulfonic and ferulic acids: DFT investigations and molecular docking studies
JS Al-Otaibi, YS Mary, YS Mary, CY Panicker… - Journal of Molecular …, 2019 - Elsevier
Cocrystals of pyrazinamide with p-toluenesulfonic acid (PZTSA) and ferulic acid (PZFER)
are investigated by density functional calculations to find geometrical parameters …
are investigated by density functional calculations to find geometrical parameters …
Hybrid and bioactive cocrystals of pyrazinamide with hydroxybenzoic acids: detailed study of structure, spectroscopic characteristics, other potential applications and …
JS Al-Otaibi, YS Mary, S Armaković… - Journal of Molecular …, 2020 - Elsevier
Three cocrystals of pyrazinamide (PYZ) with 2, 4-dihydroxy benzoic acid (2, 4HBA-PYZ), 2, 6-
dihydroxybenzoic acid (2, 6HBA-PYZ) and 3, 5-dihydroxybenzoic acid (3, 5HBA-PYZ) are …
dihydroxybenzoic acid (2, 6HBA-PYZ) and 3, 5-dihydroxybenzoic acid (3, 5HBA-PYZ) are …
Solid phase drug-drug pharmaceutical co-crystal formed between pyrazinamide and diflunisal: Structural characterization based on terahertz/Raman spectroscopy …
X Wu, Y Wang, J Xue, J Liu, J Qin, Z Hong… - Spectrochimica Acta Part A …, 2020 - Elsevier
Both pretty low solubility and high membrane permeability of diflunisal (DIF) would affect
significantly its oral bioavailability as a typical non-steroidal anti-inflammatory substance …
significantly its oral bioavailability as a typical non-steroidal anti-inflammatory substance …
First-line antituberculosis drug, pyrazinamide, its pharmaceutically relevant cocrystals and a salt
KK Sarmah, T Rajbongshi, S Bhowmick… - … Section B: Structural …, 2017 - journals.iucr.org
A few pyrazinamide (Pyz) cocrystals involving hydroxybenzoic/cinnamic acid derivatives [2,
4-dihydroxybenzoic acid (24DHBA); 2, 6-dihydroxybenzoic acid (26DHBA); 3, 5 …
4-dihydroxybenzoic acid (24DHBA); 2, 6-dihydroxybenzoic acid (26DHBA); 3, 5 …
[HTML][HTML] Pharmaceutical cocrystal formation of pyrazinamide with 3-hydroxybenzoic acid: A terahertz and Raman vibrational spectroscopies study
Q Wang, J Xue, Z Hong, Y Du - Molecules, 2019 - mdpi.com
Vibrational modes of pyrazinamide (PZA), 3-hydroxybenzoic acid (3-hBA), and their
cocrystal were characterized using terahertz time-domain (THz-TDS) and Raman vibrational …
cocrystal were characterized using terahertz time-domain (THz-TDS) and Raman vibrational …
Synthesis, co-crystal structure and characterization of pyrazinamide with m-hydroxybenzoic acid, p-hydroxybenzoic acid and 3,4-dihydroxy benzolic acid
M Lou, SH Mao, YH Luo, P Zhao, BW Sun - Research on Chemical …, 2015 - Springer
We here reported a series of co-crystal structure of pyrazinamide (PZA) with m-
hydroxybenzoic acid (MHBA), p-hydroxybenzoic acid (PHBA) and 3, 4-dihydroxy benzolic …
hydroxybenzoic acid (MHBA), p-hydroxybenzoic acid (PHBA) and 3, 4-dihydroxy benzolic …
Design, synthesis and biological activity of pyrazinamide derivatives for anti-Mycobacterium tuberculosis
S Zhou, S Yang, G Huang - Journal of Enzyme Inhibition and …, 2017 - Taylor & Francis
A total of 11 pyrazinamide derivatives were designed and synthesised using pyrazinamide
as the lead compound, which was optimised by structural modification with alkyl chains, six …
as the lead compound, which was optimised by structural modification with alkyl chains, six …
Molecular structure, spectroscopic and quantum chemical studies on benzoic acid and succinic acid co-crystals of 2-aminopyrimidine
Organic nonlinear optical co-crystals 2-aminopyrimidine benzoic acid (2APB) and 2-
aminopyrimidine succinic acid (2APS) have been successfully grown by slow solvent …
aminopyrimidine succinic acid (2APS) have been successfully grown by slow solvent …
Synthesis, Mycobacterium tuberculosis H37Rv inhibitory activity, and molecular docking study of pyrazinamide analogs
Pyrazinamide analogs 5a–h have been successfully synthesized by the Yamaguchi
esterification method with yields ranging from 6% to 86%. Among pyrazinamides 5a–h …
esterification method with yields ranging from 6% to 86%. Among pyrazinamides 5a–h …
Synthesis, Biological evaluation and molecular docking studies of new pyrazolines as an antitubercular and cytotoxic agents
BVS Lokesh, YR Prasad… - Infectious Disorders-Drug …, 2019 - ingentaconnect.com
Background: Many synthetic procedures were reported till date to prepare pyrazoline
derivatives. Some have published pyrazolines from different chalcone derivatives in the …
derivatives. Some have published pyrazolines from different chalcone derivatives in the …