In this paper, a series of novel tri (4-benzoylphenyl) phosphate derivatives with unique
precipitation-inducing properties were synthesized and used as C-terminal supports for …

To seek the novel application of organophosphorus compounds, the designed tri (4-
formylphenyl) phosphonate (TFP) derivatives were successfully synthesized herein, which …

To achieve head-to-tail cyclic peptides via the liquid-phase on-support cyclization and
synergistic self-cleavage strategy, 4, 4′-bis (diphenylphosphinyloxyl) diphenyl ketoxime …

A simple, mild, and inexpensive biphasic functionalization approach is attempted for
preparing an ideal core–shell-type resin. The core–shell-type architecture was constructed …

An efficient method for the synthesis of peptides bearing an amide at the C-terminal is
described. This method involves the attachment of a C-terminal protecting group bearing …

Since the last century, peptides have gained wide acceptance as drugs, with almost 100
already in the market and a large number in the pipeline. In this context, peptide synthesis …

Triethyl phosphate (TEP) is a new member of the Green Solid-Phase Peptide Synthesis
(GSPPS) toolbox. TEP shows almost no toxicity and no carcinogenic or mutagenic …

Amidation is the predominant reaction within the pharmaceutical setting, and it is attracting
greater attention due to the increased demand for therapeutic peptides. The high therapeutic …

Three 1-(2-nitrophenyl) ethyl-caged phospho-amino acids have been synthesized for use in
standard N α-fluorenylmethoxycarbonyl-based solid-phase peptide synthesis (SPPS). The …

The interest in developing new linkers for solid-phase peptide and organic synthesis has
increased tremendously as a result of the rapid development of combinatorial chemistry …