Synthesis and structure–antifungal activity relationships of 3-aryl-5-alkyl-2, 5-dihydrofuran-2-ones and their carbanalogues: Further refinement of tentative …

M Pour, M Špulák, V Balšánek, J Kuneš… - Bioorganic & medicinal …, 2003 - Elsevier
Two series of 3-(substituted phenyl)-5-alkyl-2, 5-dihydrofuran-2-ones related to a natural
product,(−) incrustoporine, were synthesized and their in vitro antifungal activity evaluated …

3-Phenyl-5-methyl-2H, 5H-furan-2-ones: tuning antifungal activity by varying substituents on the phenyl ring

M Pour, M Špulák, V Balšánek, J Kuneš… - Bioorganic & medicinal …, 2000 - Elsevier
A series of racemic 3-phenyl-5-methyl-2H, 5H-furan-2-ones related to a natural product,(−)
incrustoporine, was synthesized, and their antifungal activity evaluated. The key structural …

3-Phenyl-5-acyloxymethyl-2H,5H-furan-2-ones:  Synthesis and Biological Activity of a Novel Group of Potential Antifungal Drugs

M Pour, M Špulák, V Buchta, P Kubanová… - Journal of medicinal …, 2001 - ACS Publications
3-(Substituted phenyl)-5-acyloxymethyl-2 H, 5 H-furan-2-ones related to the natural product
(−) incrustoporine were synthesized and their in vitro antifungal activity evaluated. The …

Synthesis and Antifungal Activity Evaluation of 3-Hetaryl-2,5-dihydrofuran-2-ones. An Unusual Fragmentation of the Oxazole Ring via 2,3-Selenoxide Shift

J Kuneš, V Balšánek, M Pour… - … of Czechoslovak chemical …, 2001 - cccc.uochb.cas.cz
In continuing the studies on the synthesis and evaluation of antifungal activity of the
analogues of (-) incrustoporine, the replacement of the phenyl moiety at C3 of the furanone …

Stereoselective synthesis and antimicrobial activity of benzofuran-based (1E)-1-(piperidin-1-yl)-N2-arylamidrazones

HA Abdel-Aziz, AAI Mekawey - European journal of medicinal chemistry, 2009 - Elsevier
The reaction of 2-oxo-N-arylpropanehydrazonoyl chlorides 3a–e with 3-methyl-2-
benzofurancarboxylic acid hydrazide (7) furnished N-(aryl) propanehydrazonoyl chlorides …

In vitro antifungal activities of a series of dication-substituted carbazoles, furans, and benzimidazoles

M Del Poeta, WA Schell, CC Dykstra… - Antimicrobial agents …, 1998 - Am Soc Microbiol
Aromatic dicationic compounds possess antimicrobial activity against a wide range of
eucaryotic pathogens, and in the present study an examination of the structures-functions of …

Synthesis and evaluation of novel 3a, 9a-dihydro-1-ethoxycarbonyl-1-cyclopenteno [5, 4-b] benzopyran-4-ones as antifungal agents

R Goel, V Sharma, A Budhiraja, MPS Ishar - Bioorganic & medicinal …, 2012 - Elsevier
An efficient synthesis of novel antifungal 3a, 9a-dihydro-1-ethoxycarbonyl-1-cyclopenteno
[5, 4-b] benzopyran-4-ones (10a–j) through 1, 3-dipolar cycloaddition of all carbon 1, 3 …

Synthesis and antifungal activity of terpenyl-1, 4-naphthoquinone and 1, 4-anthracenedione derivatives

MÁ Castro, AM Gamito, V Tangarife-Castaño… - European Journal of …, 2013 - Elsevier
The antifungal evaluation of twenty seven simple and heterocycle-fused prenyl-1, 4-
naphthoquinones and 1, 4-anthracenediones was performed in vitro against human …

Natural products as sources of new fungicides (I): synthesis and antifungal activity of acetophenone derivatives against phytopathogenic fungi

YT Ma, HF Fan, YQ Gao, H Li… - Chemical biology & …, 2013 - Wiley Online Library
Several series of 45 acetophenone derivatives bearing various alkyl or benzyl substituents
were conveniently synthesized and their structures characterized by 1H and 13C NMR …

New diphenyl ethers from a fungus Epicoccum sorghinum L28 and their antifungal activity against phytopathogens

J Zhu, Z Li, H Lu, S Liu, W Ding, J Li, Y Xiong, C Li - Bioorganic Chemistry, 2021 - Elsevier
The strategy “IEMAHC”(Induction of Endophyte Metabolism by Adding Host Components)
was applied to the fermentation of the endophytic fungus Epicoccum sorghinum L28 from …