Regioselective Synthesis of 7-(Trimethylsilylethynyl)pyrazolo[1,5-a]pyrimidines via Reaction of Pyrazolamines with Enynones

P Golubev, EA Karpova, AS Pankova… - The Journal of …, 2016 - ACS Publications
Condensation of enynones readily available from cheap starting material with
pyrazolamines provides easy access to fluorescent 7-(trimethylsilylethynyl) pyrazolo [1, 5-a] …

Novel one pot synthesis of polysubstituted pyrazolo [1, 5-a]-and imidazo [1, 2-a] pyrimidines

AS Kiselyov, L Smith II - Tetrahedron letters, 2006 - Elsevier
We have described a convenient regioselective one-pot approach to pyrazolo [1, 5-a]-and
imidazo [1, 2-a] pyrimidine derivatives from α, β-unsaturated imines generated in situ and …

[HTML][HTML] New one-pot synthesis of 4-arylpyrazolo [3, 4-b] pyridin-6-ones based on 5-aminopyrazoles and azlactones

VY Shuvalov, EY Vlasova… - Beilstein Journal of …, 2023 - beilstein-journals.org
An effective one-pot strategy was developed for the synthesis of 4-arylpyrazolo [3, 4-b]
pyridin-6-ones from pyrazolo [3, 4-b] pyridin-6-ones, obtained by reacting 5-aminopyrazoles …

Three‐component synthesis of arene‐linked pyrazolo[1,5‐a]pyrimidines

AAM Ahmed, AEM Mekky… - Journal of Heterocyclic …, 2023 - Wiley Online Library
In this study, we aimed to establish an efficient method for synthesizing two new series of
arene‐linked pyrazolo [1, 5‐a] pyrimidines. This was achieved by reacting 1 H‐pyrazole‐3, 5 …

A mild method for the synthesis of bis-pyrazolo [3, 4-b: 4′, 3′-e] pyridine derivatives

R Qiu, S Qiao, B Peng, J Long, G Yin - Tetrahedron letters, 2018 - Elsevier
A mild and efficient method for the synthesis of bispyrazolo [3, 4-b: 4′, 3′-e] pyridines from
5-aminopyrazoles and aromatic aldehydes using an inexpensive FeCl 3 catalyst is reported …

Regioselective transition-metal-free synthesis of 2-(trimethylsilylmethylene) pyrrol-3-ones by thermal cyclization of acetylenic enamines

PR Golubev, AS Pankova… - The Journal of Organic …, 2015 - ACS Publications
Acetylenic enamines generated in situ from readily available enynones and primary amines
undergo thermal cyclization in diphenyl ether providing easy access to 4-aryl-2 …

A four-component synthesis of novel spiro [pyrazoloquinoline-oxindoles] under solvent-free conditions

H Hosseinjani-Pirdehi, K Rad-Moghadam… - Tetrahedron, 2014 - Elsevier
A domino reaction for the rapid and diverse synthesis of spiro [1 H-pyrazolo [3, 4-b] benzo [h]
dihydroquinolin-4, 3-indolin-2-ones] is reported. The synthesis represents a …

One-pot, multicomponent route to pyrazoloquinolizinones

VA Chebanov, VE Saraev, SM Desenko… - Organic …, 2007 - ACS Publications
An efficient synthesis of 5a-hydroxy-4, 5, 5a, 6, 7, 8-hexahydropyrazolo [4, 3-c] quinolizin-9-
ones based on the three-component condensation of 5-aminopyrazoles, aromatic …

NOVEL INTRAMOLECULAR CYCLIZATION OF PYRAZOLONE KETENE S,N-ACETALS FOR THE CONSTRUCTION OF METHYLSULFANYLPYRAZOLO- [4,3-b] …

GH Elgemeie, AM Elzanate… - Synthetic …, 2002 - Taylor & Francis
ABSTRACT A novel and efficient method for the synthesis of 6-substituted-7, 7a-dihydro-1,
7a-dimethyl-7-imino-2-phenyl-1 H-pyrazolo [4, 3-b] pyridin-3 (2 H)-ones via the reaction of 4 …

An efficient synthesis of fully substituted pyrazolo [3, 4-b] pyridin-5-amines from α-azidochalcones

M Adib, F Peytam - Tetrahedron, 2018 - Elsevier
A facile, mild and efficient procedure for the synthesis of fully substituted pyrazolo [3, 4-b]
pyridin-5-amines is reported. A mixture of an α-azidochalcone, a 5-aminopyrazole and t …