Facile synthesis of new pyrazolo[4′,3′:5,6]pyrano[2,3-d]pyrimidin-5(1H)-ones via the tandem intramolecular Pinner–Dimroth rearrangement and their antibacterial …

N Dorostkar-Ahmadi, A Davoodnia… - … für Naturforschung B, 2019 - degruyter.com
Abstract Some new 7-alkyl-4, 6-dihydropyrazolo [4′, 3′: 5, 6] pyrano [2, 3-d] pyrimidin-5 (1
H)-ones were prepared through heterocyclization of 6-amino-1, 4-dihydropyrano [2, 3-c] …

One-pot synthesis and antibacterial activities of pyrazolo [4′, 3′: 5, 6] pyrido [2, 3-d] pyrimidine-dione derivatives

A Bazgir, MM Khanaposhtani, AA Soorki - Bioorganic & medicinal …, 2008 - Elsevier
A one-pot and efficient method for the synthesis of pyrazolo [4′, 3′: 5, 6] pyrido [2, 3-d]
pyrimidine-dione derivatives by condensation reaction of barbituric acids, 1H-pyrazol-5 …

A Facile One-pot Synthesis of 1-Arylpyrazolo [3, 4-d] pyrimidin-4-ones

X Zhang, Q Lin, P Zhong - Molecules, 2010 - mdpi.com
One pot synthesis of 1-arylpyrazolo [3, 4-d] pyrimidin-4-ones by the reaction of 5-amino-N-
substituted-1 H-pyrazole-4-carbonitrile with different lower aliphatic acids in the presence of …

Design, synthesis, and antimicrobial activity of some new pyrazolo[3,4‐d]pyrimidines

SM Abdel‐Gawad, MM Ghorab… - … Journal of Main …, 2003 - Wiley Online Library
Benzyl‐and 2‐aryloxymethyl‐3‐amino‐1‐phenyl‐pyrazolo [3, 4‐d] pyrimidine‐4‐ones 5a–f
have been synthesized by reacting the corresponding arylacetylamino derivatives 3a–f with …

An efficient synthesis of pyrazolo[1,5-a]pyrimidines and evaluation of their antimicrobial activity

S Deshmukh, K Dingore, V Gaikwad… - Journal of Chemical …, 2016 - Springer
A series of new pyrazolo [1, 5-a] pyrimidine derivatives has been synthesized by using 7-
hydrazinyl-5-methylpyrazolo [1, 5-a] pyrimidine-3-carbonitrile 1 and 7-amino-5 …

Synthesis and antimicrobial activity of some new pyrazolo [3, 4-d] pyrimidines and thiazolo [4, 5-d] pyrimidines

JD Akbari, KB Mehta, SJ Pathak, HS Joshi - 2008 - nopr.niscpr.res.in
The desired fused ring system 3-isopropyl-4-aryl-1, 4, 5, 7-tetrahydropyrazolo [3, 4-d]
pyrimidin-6-ones 4a-d have been synthesized by the reaction of 5-isopropyl-2, 4-dihydro-3 …

[PDF][PDF] Synthesis and biological screening of some novel pyrazolo [3', 4': 4, 5] thieno [2, 3-d] pyrimidin-8-ones via a Gewald reaction

SJ Vaghasiya, DK Dodiya, AR Trivedi, VH Shah - Arkivoc, 2008 - arkat-usa.org
A new synthetic route is proposed for the synthesis of 3, 6-dimethyl-6-aryl-1, 5, 6, 7-
tetrahydro-8H-pyrazolo [3', 4': 4, 5] thieno [2, 3-d] pyrimidin-8-ones 3a-h from 5-amino-3 …

Synthesis of New Polyheterocyclic Ring Systems Derived from 3-Amino-5-bromo-4, 6-dimethyl-1H-pyrazolo [3, 4-b] pyridine

E Abdel-Latif, FS Mehdhar… - Polycyclic Aromatic …, 2019 - Taylor & Francis
Amino-5-bromo-4, 6-dimethyl-1H-pyrazolo [3, 4-b] pyridine (2) was utilized as a precursor for
the construction of new polyheterocyclic ring systems. It reacted with 4-substituted arylidene …

A regioselective synthesis of some new pyrazol-1′-ylpyrazolo [1, 5-a] pyrimidines in aqueous medium and their evaluation as antimicrobial agents

R Aggarwal, G Sumran, N Garg, A Aggarwal - European journal of …, 2011 - Elsevier
An efficient and environmental benign regioselective synthesis of some new pyrazol-1′-
ylpyrazolo [1, 5-a] pyrimidines (7b–h) has been accomplished via treatment of 3 (5)-amino-5 …

One-pot synthesis and antiproliferative evaluation of pyrazolo [3, 4-d] pyrimidine derivatives

YY Huang, LY Wang, CH Chang, YH Kuo, K Kaneko… - Tetrahedron, 2012 - Elsevier
An efficient one-pot methodology for the synthesis of pyrazolo [3, 4-d] pyrimidines was
developed by using 5-aminopyrazoles with formamide in presence of PBr3 as the coupling …