Effect of formulation variables and gamma sterilization on transcorneal permeation and stability of proniosomal gels as ocular platforms for antiglaucomal drug

S Sayed, M Abdelmoteleb, MM Amin… - AAPS PharmSciTech, 2020 - Springer
This study aims to evaluate the effect of different formulation variables (surfactant type and
HLB value) adopting full factorial design (5 1. 2 1) using coacervation phase technique on in …

Ocular ketoconazole-loaded proniosomal gels: formulation, ex vivo corneal permeation and in vivo studies

GA Abdelbary, MM Amin, MY Zakaria - Drug delivery, 2017 - Taylor & Francis
Context: Vesicular drug carriers for ocular delivery have gained a real potential.
Proniosomal gels as ocular drug carriers have been proven to be an effective way to …

Sustained ocular delivery of Dorzolamide-HCl via proniosomal gel formulation: in-vitro characterization, statistical optimization, and in-vivo pharmacodynamic …

NH Fouda, RT Abdelrehim, DA Hegazy, BA Habib - Drug delivery, 2018 - Taylor & Francis
Glaucoma is the second cause of blindness worldwide. Frequent administration of traditional
topical dosage forms may lead to patient incompliance and failure of treatment. Our study …

Development of loteprednol etabonate-loaded cationic nanoemulsified in-situ ophthalmic gel for sustained delivery and enhanced ocular bioavailability

N Patel, H Nakrani, M Raval, N Sheth - Drug delivery, 2016 - Taylor & Francis
A novel cationic nanoemulsified in-situ ophthalmic gel of loteprednol etabonate (LE) was
developed to improve the permeability and retention time of formulations for overall …

Development of dorzolamide hydrochloride in situ gel nanoemulsion for ocular delivery

HO Ammar, HA Salama, M Ghorab… - Drug development and …, 2010 - Taylor & Francis
Background: Several in situ gel-forming systems have been developed to prolong the
precorneal residence time of a drug and to improve ocular bioavailability. Poloxamer 407 …

Formulation and development of ophthalmic in situ gel for the treatment ocular inflammation and infection using application of quality by design concept

N Patel, V Thakkar, V Metalia, L Baldaniya… - Drug development …, 2016 - Taylor & Francis
Context: The conventional liquid ophthalmic delivery systems exhibit short pre-corneal
residence time and the relative impermeability to the cornea which leads to poor ocular …

Design, formulation and evaluation of carboxy methyl tamarind based in situ gelling ophthalmic drug delivery system of dorzolamide hydrochloride

FS Dasankoppa, S Kujur, HPNA Sholapur… - Indian Journal of …, 2016 - journals.lww.com
Materials and Methods: In the present investigation, an attempt has been made to design,
formulate, and evaluate in situ gelling-based ophthalmic drug delivery system dorzolamide …

Influence of hydroxypropylmethylcellulose and poloxamer composite on developed ophthalmic in situ gel: Ex vivo and in vivo characterization

R Barse, C Kokare, A Tagalpallewar - Journal of Drug Delivery Science and …, 2016 - Elsevier
The present study was planned to investigate the effect of polymer composites HPMC K15 M
and poloxamer 407 on developed dorzolamide hydrochloride in situ gel. Formulations were …

Formulation and optimization of cationic nanoemulsions for enhanced ocular delivery of dorzolamide hydrochloride using Box-Behnken design: In vitro and in vivo …

AA Kassem, A Salama, AM Mohsen - Journal of Drug Delivery Science and …, 2022 - Elsevier
The present study was designed to develop dorzolamide HCl (DRZ) loaded cationic
nanoemulsions (CNEs) for enhanced ocular delivery. CNEs were prepared employing high …

[PDF][PDF] Design, development and evaluation of cationic guar and hydroxypropyl guar based in-situ gels for ophthalmic drug delivery

FS Dasankoppa, NG Swamy - Indian Drugs, 2013 - researchgate.net
The poor bioavailability and therapeutic response exhibited by the conventional eye drops
due to rapid corneal loss is overcome by the use of ion-activated gel forming systems that …