[HTML][HTML] Antiproliferative activity of thiazole and oxazole derivatives: A systematic review of in vitro and in vivo studies

NY Guerrero-Pepinosa, MC Cardona-Trujillo… - Biomedicine & …, 2021 - Elsevier
Thiazole and oxazole are compounds with a heterocyclic nucleus that have attracted the
attention of medicinal chemistry due to the great variety of biological activities that they …

Thiazole ring—A biologically active scaffold

A Petrou, M Fesatidou, A Geronikaki - Molecules, 2021 - mdpi.com
Background: Thiazole is a good pharmacophore nucleus due to its various pharmaceutical
applications. Its derivatives have a wide range of biological activities such as antioxidant …

An overview of the synthesis and antimicrobial, antiprotozoal, and antitumor activity of thiazole and bisthiazole derivatives

AM Borcea, I Ionuț, O Crișan, O Oniga - Molecules, 2021 - mdpi.com
Thiazole, a five-membered heteroaromatic ring, is an important scaffold of a large number of
synthetic compounds. Its diverse pharmacological activity is reflected in many clinically …

Bioactive thiazole and benzothiazole derivatives

A Rouf, C Tanyeli - European journal of medicinal chemistry, 2015 - Elsevier
The heterocycles are the versatile compounds existing in almost all natural products and
synthetic organic compounds, usually associated with one or the other biological activity …

Synthetic and medicinal perspective of fused-thiazoles as anticancer agents

S Pawar, K Kumar, MK Gupta… - Anti-Cancer Agents in …, 2021 - ingentaconnect.com
Background: Cancer is second leading disease after cardiovascular disease. Presently,
Chemotherapy, Radiotherapy and use of chemicals are some treatments available these …

Recent patents on thiazole derivatives endowed with antitumor activity

R Morigi, A Locatelli, A Leoni… - Recent patents on anti …, 2015 - ingentaconnect.com
Cancer is a disease of remarkable importance in the world today and is projected to become
the primary cause of death within the coming years, therefore the design and development …

[PDF][PDF] Thiazoles: a valuable insight into the recent advances and biological activities

N Siddiqui, MF Arshad, W Ahsan… - Int. J. Pharm. Sci. Drug …, 2009 - researchgate.net
Thiazoles displayed broad range of biological activities and found in many potent
biologically active molecules such as Sulfathiazol (antimicrobial drug), Ritonavir …

2-substituted benzothiazoles as antiproliferative agents: Novel insights on structure-activity relationships

A Ammazzalorso, S Carradori, R Amoroso… - European Journal of …, 2020 - Elsevier
Given the wide spectrum of biological activities, benzothiazoles represent privileged
scaffolds in medicinal chemistry, useful in drug discovery programs to modulate biological …

Therapeutic advancement of benzothiazole derivatives in the last decennial period

S Tariq, P Kamboj, M Amir - Archiv der Pharmazie, 2019 - Wiley Online Library
Benzothiazole, a fused heterocyclic moiety, has attracted synthetic and medicinal chemists
for good reasons. It is a valuable scaffold that possesses diverse biological activities, such …

Thiazoles: having diverse biological activities

SJ Kashyap, VK Garg, PK Sharma, N Kumar… - Medicinal Chemistry …, 2012 - Springer
In the last few decades, a lot of work has been done on thiazole ring to find new compounds
related to this scaffold to act as antioxidant, analgesic, anti-inflammatory, antimicrobial …