In order to find the new potent CK2 inhibitors the 60 derivatives of 2-aminopyrimidinone and
their 6-aza-substituted analogs were synthesized and tested in vitro. Among them, the most …

Structually related to the known CK2 inhibitors, 2, 6‐disubstituted pyrazine and 4, 6‐
disubstituted pyrimidine derivatives were synthesized and their inhibitory activities toward …

A new series of furan embelin derivatives was synthesized and characterized as ATP-
competitive CK2 inhibitors. The new compounds were efficiently synthesized using a …

In this work, we describe the design, synthesis, and structure-activity relationship of 6-
(tetrazol-5-yl)-7-aminoazolo [1, 5-a] pyrimidines as inhibitors of Casein kinase 2 (CK2). At …

Identification of new small molecules inhibiting protein kinase CK2 is highly required for the
study of this protein's functions in cell and for the further development of novel …

Abstract N-Sulfonyl-N'-benzimidazol-2-yl acetamidines have been designed as CK1
inhibitors. Binding modes in the ATP pocket of CK1δ were determined by molecular …

Two classes of modified analogs of 4-(thiazol-5-yl) benzoic acid-type CK2 inhibitors were
designed. The azabenzene analogs, pyridine-and pyridazine-carboxylic acid derivatives …

A new series of 2-amino-4-phenyl-6-hydroxy-7-alkyl-pyranobenzoquinones was
synthesized as ATP-competitive CK2 inhibitors. They were readily synthesized through a …

A series of purines have been synthesized and the compounds have been tested for their
inhibitory activity against CK2. Some of them have shown an interesting activity …

An extension of our previous research work has resulted in a number of new ATP-
competitive CK2 inhibitors that have been identified among 4-aminothieno [2, 3-d] …