Late‐stage BODIPY diversification of structurally complex amino acids and peptides was
accomplished by racemization‐free palladium‐catalyzed C (sp3)− H activation …

Methods for the chemoselective modification of amino acids and peptides are powerful
techniques in biomolecular chemistry. Among other applications, they enable the total …

Spectral Dispersion and Water Solubilization of BODIPY Dyes via Palladium-Catalyzed C−H
Functionalization | Organic Letters ACS ACS Publications C&EN CAS Find my institution …

Bioorthogonal late‐stage diversification of structurally complex peptides bears enormous
potential for drug discovery and molecular imaging, among other applications. Herein, we …

Bioorthogonal late‐stage diversification of structurally complex peptides has enormous
potential for drug discovery and molecular imaging. In recent years, transition‐metal …

A highly efficient palladium-catalyzed direct C–H functionalization/annulation of BODIPYs
with alkynes has been developed for the first time to construct a series of unsymmetrical …

Modification of the aliphatic residues without an apparent functional handle has attracted
broad attention, and the scientists anticipate that the C (sp3)–H functionalizations could be …

Modification of peptides via late-stage C–H activation is an emerging strategy to construct
bioactive peptidomimetic libraries with expanded structural diversity for drug discovery …

Abstract Secondary C (sp3)− H arylations were accomplished by palladium catalysis with
triazoles as peptide bond isosteres. The unique power of this approach is highlighted by the …

The diversification of the BODIPY scaffold has been hindered by its controversial
adaptability to solid-phase chemistry. Herein we report the first solid-phase synthesis of a …