Copper-catalyzed remote CH monofluoromethylation of 8-aminoquinolines with dimethyl phosphonate as reductant

S Han, Q Wu, L Mele, L Ding, J Li, D Zou, Y Wu, Y Wu - Tetrahedron Letters, 2019 - Elsevier
A simple and efficient copper-catalyzed monofluoromethylation of 8-aminoquinolines with 2-
bromo-2-fluoroacetate has been described with HPO (OMe) 2 (dimethyl phosphonate) as …

Copper‐Catalyzed Aryltrifluoromethylation of N‐Phenylcinnamamides: Access to Trifluoromethylated 3,4‐Dihydroquinolin‐2(1 H)‐ones

Q Wang, G Han, Y Liu, Q Wang - Advanced Synthesis & …, 2015 - Wiley Online Library
Copper‐Catalyzed Aryltrifluoromethylation of N‐Phenylcinnamamides: Access to
Trifluoromethylated 3,4‐Dihydroquinolin‐2(1 H)‐ones - Wang - 2015 - Advanced Synthesis & …

Copper-catalyzed remote CH ethoxycarbonyldifluoromethylation of 8-aminoquinolines with bis (pinacolato) diboron as reductant

S Han, A Liang, X Ren, X Gao, J Li, D Zou, Y Wu… - Tetrahedron letters, 2017 - Elsevier
A simple protocol for the copper/B 2 pin 2-catalyzed Csingle bondH
ethoxycarbonyldifluoromethylation of 8-aminoquinoline scaffolds with functionalized …

Oxidative Remote C− H Trifluoromethylation of Quinolineamides on the C5 Position with Iodobenzene Diacetate as the Oxidizing Agent

Z Wu, Y He, C Ma, X Zhou, X Liu, Y Li… - Asian Journal of …, 2016 - Wiley Online Library
A facile, metal‐free protocol has been developed for the remote trifluoromethylation of 8‐
aminoquinoline scaffolds on the C5 position, which is difficult to functionalize. In this method …

Copper-mediated C–H trifluoromethylation of quinones

NO Ilchenko, PG Janson, KJ Szabó - Chemical Communications, 2013 - pubs.rsc.org
Copper-mediated C–H trifluoromethylation of quinones - Chemical Communications (RSC
Publishing) DOI:10.1039/C3CC43357A Royal Society of Chemistry View PDF VersionPrevious …

5-Position-selective C–H trifluoromethylation of 8-aminoquinoline derivatives

Y Kuninobu, M Nishi, M Kanai - Organic & Biomolecular Chemistry, 2016 - pubs.rsc.org
We developed a copper-catalyzed 5-position-selective C–H trifluoromethylation of 8-
aminoquinoline derivatives. The reaction proceeded with high functional group tolerance …

Ruthenium‐Catalyzed Difluoroalkylation of 8‐Aminoquinoline Amides at the C5‐Position

C Chen, R Zeng, J Zhang… - European Journal of …, 2017 - Wiley Online Library
A ruthenium‐catalyzed highly selective difluoromethylation of 8‐aminoquinoline amides at
the C5 position has been developed. It tolerates a broad range of functional groups …

Nickel-catalyzed C–H bond trifluoromethylation of 8-aminoquinoline derivatives by acyl-directed functionalization

X Liu, G Mao, J Qiao, C Xu, H Liu, J Ma… - Organic Chemistry …, 2019 - pubs.rsc.org
A Ni (TFA) 2-catalyzed ortho-trifluoromethylation of 8-aminoquinoline derivatives was
developed by acyl-directed C–H functionalization. A series of 7-trifluoromethylquinolinamine …

Copper-Catalyzed Direct C–H Trifluoromethylation of Quinones

X Wang, Y Ye, G Ji, Y Xu, S Zhang, J Feng… - Organic …, 2013 - ACS Publications
Copper-Catalyzed Direct C–H Trifluoromethylation of Quinones | Organic Letters ACS ACS
Publications C&EN CAS Find my institution Log In Organic Letters ACS Publications. Most …

2-Position-selective C–H perfluoroalkylation of quinoline derivatives

T Shirai, M Kanai, Y Kuninobu - Organic letters, 2018 - ACS Publications
We developed 2-position-selective, direct C–H trifluoromethylation, pentafluoroethylation,
and heptafluoropropylation of quinoline derivatives. Regioselective transformation was …