Efficient synthesis, antibacterial, antifungal, antioxidant and cytotoxicity study of 2‐(2‐hydrazineyl) thiazole derivatives
VA Adole, RA More, BS Jagdale, TB Pawar… - …, 2020 - Wiley Online Library
In the present investigation, an alluring green PEG‐400 mediated one‐pot synthesis of
novel 2‐(2‐hydrazinyl) thiazole derivatives from 1, 2, 6, 7‐tetrahydro‐8H‐indeno [5, 4‐b] …
novel 2‐(2‐hydrazinyl) thiazole derivatives from 1, 2, 6, 7‐tetrahydro‐8H‐indeno [5, 4‐b] …
Design, synthesis and biological evaluation of new series of benzotriazole-pyrazole clubbed thiazole hybrids as bioactive heterocycles: Antibacterial, antifungal …
KB Gangurde, RA More, VA Adole… - Journal of Molecular …, 2024 - Elsevier
The need for novel heterocyclic compounds with robust biological action is a result of the
emergence of numerous pandemics and microbial resistance. To search antibacterial and …
emergence of numerous pandemics and microbial resistance. To search antibacterial and …
[HTML][HTML] Design, synthesis and docking studies of new hydrazinyl-thiazole derivatives as anticancer and antimicrobial agents
Increase in the number of infections caused by pathogenic microbes in cancer patients has
prompted the searcher to invest in the development of agents having dual anticancer and …
prompted the searcher to invest in the development of agents having dual anticancer and …
A facile access and evaluation of some novel thiazole and 1, 3, 4-thiadiazole derivatives incorporating thiazole moiety as potent anticancer agents
Background Many heterocyclic compounds containing thiazole or 1, 3, 4-thiadiazole ring in
their skeletons have been reported to possess various pharmacological activities especially …
their skeletons have been reported to possess various pharmacological activities especially …
Synthesis, anti-inflammatory and antimicrobial evaluation of novel 1-acetyl-3, 5-diaryl-4, 5-dihydro (1H) pyrazole derivatives bearing urea, thiourea and sulfonamide …
AP Keche, GD Hatnapure, RH Tale, AH Rodge… - Bioorganic & medicinal …, 2012 - Elsevier
A series of novel 1-acetyl-3-(3, 4-dimethoxypheny)-5-(4-(3-(arylureido/arylthioureido/
arylsulfonamido) phenyl)-4, 5-dihydropyrazole derivatives of biological interest have been …
arylsulfonamido) phenyl)-4, 5-dihydropyrazole derivatives of biological interest have been …
Synthesis, X-ray crystallographic, spectroscopic and computational studies of aminothiazole derivatives
Aminothiazole organic compounds have diverse biological applications. Herein we report
the synthesis of two aminothiazole derivatives: 4-(biphenyl-4-yl) thiazol-2-amine (1) and 4 …
the synthesis of two aminothiazole derivatives: 4-(biphenyl-4-yl) thiazol-2-amine (1) and 4 …
Synthesis, molecular docking study, and cytotoxicity evaluation of some novel 1, 3, 4-thiadiazole as well as 1, 3-thiazole derivatives bearing a pyridine moiety
Pyridine, 1, 3, 4-thiadiazole, and 1, 3-thiazole derivatives have various biological activities,
such as antimicrobial, analgesic, anticonvulsant, and antitubercular, as well as other …
such as antimicrobial, analgesic, anticonvulsant, and antitubercular, as well as other …
Exploring of antioxidant and antibacterial properties of novel 1, 3, 4-thiadiazole derivatives: Facile synthesis, structural elucidation and DFT approach to antioxidant …
In recent years, compounds containing thiophene and 1, 3, 4-thiadiazole skeletons have
become important cyclic compounds, especially in medicinal chemistry. In this manner, we …
become important cyclic compounds, especially in medicinal chemistry. In this manner, we …
Synthesis, antibacterial activity and quantum-chemical studies of novel 2-arylidenehydrazinyl-4-arylthiazole analogues
MS Alam, L Liu, YE Lee, DU Lee - Chemical and Pharmaceutical …, 2011 - jstage.jst.go.jp
A new series of 2-arylidenehydrazinyl-4-arylthiazole derivatives (2a—k) was designed and
synthesized through a rapid, simple, and efficient methodology in excellent isolated yield …
synthesized through a rapid, simple, and efficient methodology in excellent isolated yield …
Design, synthesis, characterization, in vitro screening, molecular docking, 3D-QSAR, and ADME-Tox investigations of novel pyrazole derivatives as antimicrobial …
M Chalkha, M Akhazzane, FZ Moussaid… - New Journal of …, 2022 - pubs.rsc.org
In this work, we report the synthesis of some new pyrazole derivatives via an efficient and
practical procedure. The structures of the obtained compounds were established using …
practical procedure. The structures of the obtained compounds were established using …