Mn-and Co-catalyzed aminocyclizations of unsaturated hydrazones providing a broad range of functionalized pyrazolines

M Balkenhohl, S Kölbl, T Georgiev, EM Carreira - JACS Au, 2021 - ACS Publications
Manganese-and cobalt-catalyzed aminocyclization reactions of unsaturated hydrazones are
reported. Whereas manganese catalysis provides access to pyrazoline and …

An overview on synthesis and biological activity of chalcone derived pyrazolines

A Tiwari, A Bendi, AS Bhathiwal - ChemistrySelect, 2021 - Wiley Online Library
Chalcones are α, β unsaturated aromatic ketones having enone moiety and exhibit a wide
array of pharmaceutical and biological activities. Chalcones possess a wide range of …

Synthesis of thymol-based pyrazolines: An effort to perceive novel potent-antimalarials

DS Raghuvanshi, N Verma, SV Singh, S Khare… - Bioorganic …, 2019 - Elsevier
A series of thymol based substituted pyrazolines and chalcones was synthesized and
evaluated for antimalarial activity, using in-vitro and in-vivo malaria models. All the target …

Synthesis of 1, 3, 5-trisubstituted pyrazoles via 1, 3-dipolar cycloaddition of nitrile imines with ninhydrin-derived Morita–Baylis–Hillman carbonates

KK Wang, YL Li, J Jing, R Chen, NN Zhao… - Organic & …, 2022 - pubs.rsc.org
An effective synthetic method for 1, 3, 5-trisubstituted pyrazoles via 1, 3-dipolar cycloaddition
reaction has been developed. This reaction could smoothly proceed between ninhydrin …

PEG-mediated synthesis, antibacterial, antifungal and antioxidant studies of some new 1, 3, 5-trisubstituted 2-pyrazolines

SL Dhonnar, BS Jagdale, VA Adole, NV Sadgir - Molecular Diversity, 2023 - Springer
Abstract A new series of 1, 3, 5-trisubstituted 2-pyrazoline derivatives (3a–l) are synthesized
in good to excellent yields from the corresponding chalcones (1a–h) and acid hydrazides …

Antibacterial potential of chalcones and its derivatives against Staphylococcus aureus

L da Silva, IA Donato, CAC Gonçalves, JR Scherf… - 3 Biotech, 2023 - Springer
Chalcones are natural substances found in the metabolism of several botanical families.
Their structure consists of 1, 3-diphenyl-2-propen-1-one and they are characterized by …

Unveiling the Substituent Effects in the Stereochemistry of [3+ 2] Cycloaddition Reactions of Aryl‐and Alkyldiazomethylphosphonates with Norbornadiene within a …

LR Domingo, N Acharjee - ChemistrySelect, 2021 - Wiley Online Library
Abstract The [3+ 2] cycloaddition (32CA) reactions of norbornadiene with aryl and alkyl
substituted diazomethylphosphonates (SDAPs) have been studied within the molecular …

[HTML][HTML] Chloramine-T (N-chloro-p-toluenesulfonamide sodium salt), a versatile reagent in organic synthesis and analytical chemistry: An up to date review

YN Nayak, SL Gaonkar, EAM Saleh… - Journal of Saudi …, 2022 - Elsevier
Abstract Chloramine-T (CAT), the sodium salt of N-chloro-p-toluenesulfonamide, is a low-
cost mild oxidizing agent with a wide range of uses. Most importantly, it can be used in …

Synthesis and characterization of some new pyrazolines and their inhibitory potencies against carbonic anhydrases

G Çelik, T Arslan, M Şentürk, D Ekinci - Archiv der Pharmazie, 2020 - Wiley Online Library
The inhibition of the two human cytosolic carbonic anhydrase (hCA; EC 4.2. 1.1) isozymes I
and II with some new pyrazoline derivatives was investigated for the first time. The structures …

In‐situ Utilization of Non‐Stabilized Diazoalkanes from (3+2) Cycloaddition of Linear N,N‐Disilyl Enamines and Azides

V Do Cao, S Lee, S Joung - Advanced Synthesis & Catalysis, 2024 - Wiley Online Library
Abstract A (3+ 2) cycloaddition reaction of linear N, N‐disilyl enamines and organic azides is
investigated. The N, N‐disilyl enamines, derived from the selective double hydrosilylation of …