1, 3, 4-Oxadiazole containing compounds as therapeutic targets for cancer therapy
MJ Ahsan - Mini Reviews in Medicinal Chemistry, 2022 - ingentaconnect.com
Background: Cancer is the first or second leading cause of premature death in 134 of 183
countries in the world. 1, 3, 4-Oxadiazoles are five membered heterocyclic rings containing …
countries in the world. 1, 3, 4-Oxadiazoles are five membered heterocyclic rings containing …
Synthesis, docking studies into CDK-2 and anticancer activity of new derivatives based pyrimidine scaffold and their derived glycosides
AAH Rahman, IF Nassar, AKF Shaban… - Mini Reviews in …, 2019 - ingentaconnect.com
Background & Objective: New diaryl-substituted pyrimidinedione compounds, their thioxo
derivatives as well as their bicyclic thiazole compounds were synthesized and …
derivatives as well as their bicyclic thiazole compounds were synthesized and …
Synthesis of novel 1, 2, 3-triazole based acridine and benzothiazole scaffold N-glycosides with anti-proliferative activity, docking studies, and comparative …
AM Fahim, HEM Tolan, WA El-Sayed - Journal of Molecular Structure, 2022 - Elsevier
In this investigation, the cycloaddition reaction of azide-alkyne derivatives 1a, b with
glucopyranose azide 2a, b was catalyzed via Cu (I) to afford the corresponding acetylated 1 …
glucopyranose azide 2a, b was catalyzed via Cu (I) to afford the corresponding acetylated 1 …
Synthesis and anticancer activity of new ((Furan-2-yl)-1, 3, 4-thiadiazolyl)-1, 3, 4-oxadiazole acyclic sugar derivatives
AF Kassem, IF Nassar, MT Abdel-Aal… - Chemical and …, 2019 - jstage.jst.go.jp
New sugar hydrazones incorporating furan and/or 1, 3, 4-thiadiazole ring systems were
synthesized by reaction of the corresponding hydrazide with different aldose sugars …
synthesized by reaction of the corresponding hydrazide with different aldose sugars …
[HTML][HTML] Discovery of new pyrazolopyridine, furopyridine, and pyridine derivatives as CDK2 inhibitors: Design, synthesis, docking studies, and anti-proliferative activity
AAH Abdel-Rahman, AKF Shaban, IF Nassar… - Molecules, 2021 - mdpi.com
New pyridine, pyrazoloyridine, and furopyridine derivatives substituted with naphthyl and
thienyl moieties were designed and synthesized starting from 6-(naphthalen-2-yl)-2-oxo-4 …
thienyl moieties were designed and synthesized starting from 6-(naphthalen-2-yl)-2-oxo-4 …
[HTML][HTML] Synthesis and Cytotoxic Activity of New 1,3,4-Thiadiazole Thioglycosides and 1,2,3-Triazolyl-1,3,4-Thiadiazole N-glycosides
New 1, 3, 4-thiadiazole thioglycosides linked to substituted arylidine systems were
synthesized via glycosylation of the prepared 1, 3, 4-thiadiazole thiol compounds. Click …
synthesized via glycosylation of the prepared 1, 3, 4-thiadiazole thiol compounds. Click …
Spectral studies, thermal investigations, and anticancer activity of some divalent metal complexes derived from 2‐(4‐bromophenylamino) acetohydrazide ligand
EM Emara, WA El‐Sayed… - Applied …, 2022 - Wiley Online Library
A series of biologically active metal complexes was yielded from the reactions of 2‐(4‐
bromophenylamino) acetohydrazide ligand (HL) with Co (II), Ni (II), Cu (II), Cd (II) chlorides …
bromophenylamino) acetohydrazide ligand (HL) with Co (II), Ni (II), Cu (II), Cd (II) chlorides …
Synthesis, anticancer activity and molecular docking of new triazolo[4,5-d]pyrimidines based thienopyrimidine system and their derived N-glycosides and …
RR Khattab, AA Hassan, DA A. Osman… - … Nucleotides & Nucleic …, 2021 - Taylor & Francis
A series of new substituted triazolo [4, 5-d] pyrimidine derivatives linked to thienopyrimidine
ring system were prepared as a hybrid heterocyclic systems, as possible nucleobases …
ring system were prepared as a hybrid heterocyclic systems, as possible nucleobases …
Anticancer activity of new substituted pyrimidines, their thioglycosides and thiazolopyrimidine derivatives
MNM Yousif, WA El-Sayed, HAS Abbas… - Journal of applied …, 2017 - japsonline.com
Novel functionalized pyrimidine, thioxopyrimidine, iminopyrimidine derivatives and their
derived bicyclic thiazolopyrimidine compounds were synthesized. The substituted arylidine …
derived bicyclic thiazolopyrimidine compounds were synthesized. The substituted arylidine …
Chemical and enzymatic synthesis of S-linked sugars and glycoconjugates
M Qiao, L Zhang, R Jiao, S Zhang, B Li, X Zhang - Tetrahedron, 2021 - Elsevier
S-Linked oligosaccharide/polysaccharide and glycoconjugates including glycolipid,
glycoprotein, saponin and others, in which the glycosidic oxygen is replaced by a sulfur …
glycoprotein, saponin and others, in which the glycosidic oxygen is replaced by a sulfur …