Screening for metabolically stable aryl‐propionamide‐derived selective androgen receptor modulators for doping control purposes

M Thevis, M Kamber… - Rapid Communications in …, 2006 - Wiley Online Library
Anabolic agents have been among the most frequently detected drugs in amateur and
professional sport. A novel class of therapeutics presumably complementing anabolic …

A bioisosteric approach to the discovery of indole carbinol androgen receptor ligands

JC Lanter, JJ Fiordeliso, GF Allan, A Musto… - Bioorganic & medicinal …, 2006 - Elsevier
Two potential bioisosteres of the nonsteroidal antiandrogen bicalutamide, an
imidazolidinone and an indole, were synthesized and tested for their androgen receptor …