Nonsteroidal selective androgen receptor modulators (SARMs): dissociating the anabolic and androgenic activities of the androgen receptor for therapeutic benefit
ML Mohler, CE Bohl, A Jones, CC Coss… - Journal of medicinal …, 2009 - ACS Publications
Interest in the development and therapeutic potential of nonsteroidal tissue-selective
androgen receptor modulators (SARMs) a has increased dramatically within the past …
androgen receptor modulators (SARMs) a has increased dramatically within the past …
Nonsteroidal selective androgen receptor modulator Ostarine™ in cancer cachexia
MF Zilbermint, AS Dobs - Future Oncology, 2009 - Future Medicine
Cancer cachexia is a complex syndrome, affecting up to 60% of the approximately 1.4
million patients diagnosed with cancer each year in the USA. This condition is characterized …
million patients diagnosed with cancer each year in the USA. This condition is characterized …
Detection of the arylpropionamide‐derived selective androgen receptor modulator (SARM) S‐4 (Andarine) in a black‐market product
M Thevis, H Geyer, M Kamber… - Drug testing and …, 2009 - Wiley Online Library
Non‐steroidal and tissue‐selective anabolic agents such as selective androgen receptor
modulators (SARMs) represent a promising class of therapeutics for the treatment of various …
modulators (SARMs) represent a promising class of therapeutics for the treatment of various …
Emerging drugs: mechanism of action, mass spectrometry and doping control analysis
M Thevis, A Thomas, M Kohler, S Beuck… - Journal of mass …, 2009 - Wiley Online Library
The number of compounds and doping methods in sports is in a state of constant flux. In
addition to 'traditional'doping agents, such as anabolic androgenic steroids or erythropoietin …
addition to 'traditional'doping agents, such as anabolic androgenic steroids or erythropoietin …
Doping control analysis of emerging drugs in human plasma–identification of GW501516, S‐107, JTV‐519, and S‐40503
M Thevis, S Beuck, A Thomas, B Kortner… - … Journal Devoted to …, 2009 - Wiley Online Library
An important aspect of preventive doping research is the rapid implementation of tests for
emerging drugs with potential for misuse into routine doping control assays. New …
emerging drugs with potential for misuse into routine doping control assays. New …
Recent advances in the development of selective androgen receptor modulators
X Zhang, JC Lanter, Z Sui - Expert Opinion on Therapeutic Patents, 2009 - Taylor & Francis
Background: The androgens testosterone and its more potent tissue metabolite 5-α-
dihydrotesterone regulate diverse physiological process involving both reproductive and …
dihydrotesterone regulate diverse physiological process involving both reproductive and …