Biginelli reaction: a green perspective
The Biginelli Reaction is a one-pot acid catalysed cyclocondensation of β-keto ester, urea
and aromatic aldehyde which leads to the synthesis of functionalised 3, 4-dihydro-2 (H) …
and aromatic aldehyde which leads to the synthesis of functionalised 3, 4-dihydro-2 (H) …
A CuAAC/Ullmann C–C Coupling Tandem Reaction: Copper-Catalyzed Reactions of Organic Azides with N-(2-Iodoaryl)propiolamides or 2-Iodo-N-(prop-2-ynyl) …
A novel copper-catalyzed tandem reaction was developed by utilizing two famous copper-
catalyzed reactions, CuAAC and Ullmann coupling. The trapping of the C–Cu intermediate …
catalyzed reactions, CuAAC and Ullmann coupling. The trapping of the C–Cu intermediate …
Biginelli condensation: synthesis and structure diversification of 3, 4-dihydropyrimidin-2 (1H)-one derivatives
The realization of therapeutic potential of 3, 4-dihydropyrimidin-2 (1H)-ones (DHPMs) and
their structural as well as receptor bound conformational similarity with potent cardiovascular …
their structural as well as receptor bound conformational similarity with potent cardiovascular …
One-pot synthesis of useful heterocycles in medicinal chemistry using a cascade strategy
To access useful heterocycles in medicinal chemistry such as pyridazinones,
dihydropyrimidinones, and dihydropyrimidinthiones, a “green” mild and highly efficient one …
dihydropyrimidinones, and dihydropyrimidinthiones, a “green” mild and highly efficient one …
Combining click-multicomponent reaction: one-pot synthesis of triazolyl methoxy-phenyl indazolo[2,1-b]phthalazine-trione derivatives
Abstract [(1, 2, 3-Triazol-4-yl) methoxy-phenyl]-2 H-indazolo [2, 1-b] phthalazine-trione
derivatives were synthesized in a simple and efficient method from the one-pot four …
derivatives were synthesized in a simple and efficient method from the one-pot four …
α-Azido ketones. Part 7: synthesis of 1,4-disubstituted triazoles by the “click” reaction of various terminal acetylenes with phenacyl azides or α-azidobenzo(hetera) …
K Kónya, S Fekete, A Ábrahám, T Patonay - Molecular diversity, 2012 - Springer
Abstract Copper (I)-catalyzed alkyne-azide 1, 3-cycloaddition reaction (CuAAC, Sharpless–
Meldal reaction) of various α-azido ketones such as substituted 2-azidoacetophenones, 2 …
Meldal reaction) of various α-azido ketones such as substituted 2-azidoacetophenones, 2 …
Synthesis of phenyl azides bearing (E)-2-halovinyl group
W Zhang, C Kuang, Q Yang - Research on Chemical Intermediates, 2012 - Springer
A series of phenyl azides bearing (E)-2-halovinyl groups were synthesized in high yields by
treatment of (E)-3-(4-azidophenyl)-and (E)-3-(2-azidophenyl) acrylic acid with N …
treatment of (E)-3-(4-azidophenyl)-and (E)-3-(2-azidophenyl) acrylic acid with N …
[PDF][PDF] Інститут органічної хімії НАН України, 02094, м. Київ, вул. Мурманська, 5. E mail: mvovk@ i. com. ua Ключові слова: 3, 4ЅдигідропіримідинЅ2 (1H) Ѕони; …
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[PDF][PDF] Heterocyclic scaffolds form the core of many pharmaceutically relevant substances. Not surprisingly, therefore, many publications in the area of microwave …
CO Kappe, A Stadler… - … and Principles in …, 2012 - perpus.univpancasila.ac.id
The vanadium-catalyzed epoxidation of hindered homoallylic alcohols has been described
by Prieto and coworkers [2]. The reaction times for the epoxidation in a series of cis-and …
by Prieto and coworkers [2]. The reaction times for the epoxidation in a series of cis-and …