Benzofuran derivatives: a patent review
KM Dawood - Expert opinion on therapeutic patents, 2013 - Taylor & Francis
Introduction: Benzofuran moiety constitutes the core of several interesting pharmacologically
active natural products. Benzofurans are among feasible potent active inhibitors against …
active natural products. Benzofurans are among feasible potent active inhibitors against …
[图书][B] Palladium-catalyzed coupling reactions: practical aspects and future developments
Á Molnár - 2013 - books.google.com
This handbook and ready reference brings together all significant issues of practical
importance in selected topics discussing recent significant achievements for interested …
importance in selected topics discussing recent significant achievements for interested …
Design, synthesis and structure–activity relationships of some novel, highly potent anti-invasive (E)-and (Z)-stilbenes
BI Roman, LM De Coen, STFC Mortier… - Bioorganic & medicinal …, 2013 - Elsevier
In our ongoing exploration of the structure–activity landscape of anti-invasive chalcones, we
have prepared and evaluated a number of structurally related (E)-and (Z)-stilbenes. These …
have prepared and evaluated a number of structurally related (E)-and (Z)-stilbenes. These …
Synthesis and biochemical activities of antiproliferative amino acid and phosphate derivatives of microtubule-disrupting β-lactam combretastatins
NM O'Boyle, LM Greene, NO Keely, S Wang… - European journal of …, 2013 - Elsevier
The synthesis and biochemical activities of novel water-soluble β-lactam analogues of
combretastatin A-4 are described. The first series of compounds investigated, β-lactam …
combretastatin A-4 are described. The first series of compounds investigated, β-lactam …
Synthesis, biological evaluation, and molecular modeling studies of novel heterocyclic compounds as anti-proliferative agents
Two novel series of heterocyclic compounds have been synthesized. In first series, isatin
was allowed to react with substituted aromatic/cyclic carbonyl compounds to get desired …
was allowed to react with substituted aromatic/cyclic carbonyl compounds to get desired …
BPR0C305, an orally active microtubule-disrupting anticancer agent
WT Li, TK Yeh, JS Song, YN Yang, TW Chen… - Anti-Cancer …, 2013 - journals.lww.com
BPR0C305 is a novel N-substituted indolyl glyoxylamide previously reported with in-vitro
cytotoxic activity against a panel of human cancer cells including P-gp-expressing multiple …
cytotoxic activity against a panel of human cancer cells including P-gp-expressing multiple …
Methods of detecting and treatment of cancers using Scutellaria barbata extract
I Cohen - US Patent 8,512,961, 2013 - Google Patents
(57) ABSTRACT An extract of Scutellaria Barbata D. Don is effective in the arrest of cancer
cell growth. The extract of Scutellaria Bar bata D. Don may be used as a therapeutic …
cell growth. The extract of Scutellaria Bar bata D. Don may be used as a therapeutic …
Mechanistic Studies on Regioselective Dephosphorylation of Phosphate Prodrugs during a Facile Synthesis of Antitumor Phosphorylated 2-Phenyl-6, 7 …
Phosphorylation of 2-(3-hydroxy-5-methoxyphenyl)-6, 7-methylenedioxy-1 H-quinolin-4-one
(1) afforded diphosphate 2. We found that, upon treatment with methanol under mild …
(1) afforded diphosphate 2. We found that, upon treatment with methanol under mild …
[引用][C] Palladium‐Catalyzed Cross‐Coupling Reactions–Industrial Applications
A Dumrath, C Lübbe, M Beller - Palladium‐Catalyzed Coupling …, 2013 - Wiley Online Library
This chapter contains sections titled: Introduction Suzuki–Miyaura Reactions Heck–Mizoroki
Reactions Sonogashira–Hagihara Reactions Carbonylations Cyanations Negishi Coupling …
Reactions Sonogashira–Hagihara Reactions Carbonylations Cyanations Negishi Coupling …