On DABAL-Me3 promoted formation of amides

N Dubois, D Glynn, T McInally, B Rhodes, S Woodward… - Tetrahedron, 2013 - Elsevier
The range and utility of DABAL-Me 3 couplings of methyl esters and free carboxylic acids
with primary and secondary amines under a variety of conditions (reflux, sealed tube …

An efficient one-pot microwave assisted synthesis of dibenzoazepinones

PK Deb, S Sharma, A Borude, RP Singh, D Kumar… - Tetrahedron …, 2013 - Elsevier
Microwave assisted one-pot synthesis of substituted 5H-dibenzo [b, d] azepin-6 (7H)-ones
from 2-(2-bromophenyl) acetic acid esters and 2-aminophenyl boronates has been …

[PDF][PDF] Targeting of estrogen biosynthesis and hormone receptor signalling pathways for the treatment of cancer

M Mottinelli - 2013 - purehost.bath.ac.uk
The tetrahydroisoquinoline (THIQ) core structure is explored as a steroidomimetic nucleus
with attractive pharmaceutical properties. A library was synthesised employing Pomeranz …

[引用][C] Advancing API Synthesis

C Challener - 2013 - Advanstar

[引用][C] Reducing the Complexity of Commercial-Scale Amide Formation

C Challener - 2013 - Advanstar