C–H Arylation of Heterocyclic N-Oxides Through in Situ Diazotisation Of Anilines without Added Promoters: A Green And Selective Coupling Process
AP Colleville, RAJ Horan, S Olazabal… - … Process Research & …, 2016 - ACS Publications
A green and selective method for the generation of biaryl compounds through C–H arylation
of heterocyclic N-oxides, in which the addition of ascorbic acid as a promoter is not required …
of heterocyclic N-oxides, in which the addition of ascorbic acid as a promoter is not required …
A Facile and Efficient Method for the Formation of Unsymmetrical Ureas Using DABAL-Me3
A practical synthetic method for the formation of unsymmetrical-substituted ureas is
described. The synthesis of the unsymmetrical ureas was readily performed from 2, 2, 2 …
described. The synthesis of the unsymmetrical ureas was readily performed from 2, 2, 2 …
Synthèse d'hétérocycles spiraniques à visée thérapeutique
F Magne - 2016 - theses.hal.science
Depuis quelques années, l'élaboration de molécules spiraniques connait un essor
considérable avec, en particulier, comme but essentiel l'accroissement de la diversité …
considérable avec, en particulier, comme but essentiel l'accroissement de la diversité …
Development of novel inhibitors of carbohydrate-processing targets involved in Mycobacterium tuberculosis cell wall biosynthesis
B Whitehurst - 2016 - stax.strath.ac.uk
Tuberculosis (TB) remains one of the world's most lethal infectious diseases. The
emergence and increasing prevalence of drug-resistant strains of Mycobacterium …
emergence and increasing prevalence of drug-resistant strains of Mycobacterium …
A medicinal chemistry approach towards brodomain epigenetic modulators
RP Law - 2016 - stax.strath.ac.uk
Bromodomains are a family of epigenetic reader domains which recognize acetylated
histone lysine residues, recruiting transcription factors to specific DNA locales. Aberrant …
histone lysine residues, recruiting transcription factors to specific DNA locales. Aberrant …