Synthesis, antibacterial and antifungal activities of naphthoquinone derivatives: a structure–activity relationship study

JM Sánchez-Calvo, GR Barbero… - Medicinal Chemistry …, 2016 - Springer
Abstract The synthesis of 1, 4-naphthoquinone derivatives is of great interest since these
compounds exhibit strong activity as antimalarial, antibacterial, antifungal and anticancer …

[PDF][PDF] 1, 5-Benzothiazepine: Bioactivity and targets

R Kaur, K Singh, R Singh - Chem. Biol. Lett, 2016 - researchgate.net
Benzothiazepine nucleus is present in a number of clinically used drugs such as diltiazem,
clentiazem, thiazesim, quetiapine, and clothiapine. 1, 5-Benzothiazepine can be easily …

Synthesis, antibacterial and cytotoxic activities of new biflorin-based hydrazones and oximes

LGS Souza, MCS Almeida, TLG Lemos… - Bioorganic & Medicinal …, 2016 - Elsevier
Biflorin 1 is a biologically active quinone, isolated from Capraria biflora. Five new biflorin-
based nitrogen derivatives were synthesized, of which two were mixtures of (E)-and (Z) …

[HTML][HTML] Synthesis, in vitro Antifungal Activity and Molecular Modeling Studies of New Mannich Bases Derived from Lawsone

JF Allochio Filho, LL Roldi, M Delarmelina… - Journal of the Brazilian …, 2016 - SciELO Brasil
Hydroxynaphthoquinones such as lawsone (2-hydroxy-1, 4-naphthoquinone) have proven
to be effective antifungal agents. These compounds were tested for antifungal activity …

[PDF][PDF] Synthesis, biological, and computational study of naphthoquinone derivatives containing heteroatoms

NDC Heteroatoms - J. Chem. Soc. Pak, 2016 - researchgate.net
A number of 2-(aryl/alkyl) thio-3-chloro-l, 4-naphthoquinones (3a-g) and 2, 3-(aryl/alkyl) thio-
l, 4-naphthoquinones (4a-d, 4f-g) were obtained by the reactions of 2, 3-dichloro-1, 4 …

Synthesis, antibacterial and antifungal evaluation of thio-or piperazinyl-substituted 1, 4-naphthoquinone derivatives

C Ibis, Z Ozsoy-Gunes, AF Tuyun, SS Ayla… - Journal of Sulfur …, 2016 - Taylor & Francis
ABSTRACT A series of S-, S, S-, S, O-, N-and N, S-derivatives from 2, 3-dichloro-1, 4-
naphthoquinone compound 1 were synthesized in different reaction media and evaluated …

[PDF][PDF] Screening of thioalkanoic substituted 1, 4-naphthoquinones as potent antimicrobial agents

G RĂU, FM CREŢU, A Berbecaru-Iovan… - …, 2016 - farmaciajournal.com
In the present study, there are described the synthesis and evaluation of physico-chemical
properties and antimicrobial activity of some hetero-1, 4-naphthoquinones containing thiol …

[PDF][PDF] AZOT VE KÜKÜRT İÇEREN YENİ HETERO KİNONLARIN SENTEZİ VE KARAKTERİZASYONU

S KURBAN, MÇ SAYIL, II Danışman, Z GÖKMEN - nek.istanbul.edu.tr
Ve bugünlere gelmemi sağlayan, maddi ve manevi olarak her zaman arkamda duran, tez
çalışmalarım boyunca desteğini esirgemeyen çok kıymetli eşim ve kızım Funda Kurban ve …

[引用][C] Oksijen ve kükürt sübstitüe 1, 4-naftakinonların sentezi ve antimikrobiyal aktivitelerinin incelenmesi

H Kilinç - platform.almanhal.com
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[引用][C] THIOUREA DERIVATIVES OF 4-AZATRICYCLO [5.2. 2.02, 6] UNDEC-8-ENE-3, 5-DIONE ñ SYNTHESIS AND BIOLOGICAL ACTIVITY

A BIELENICA, J STEFA—SKA, AE KOZIO, F IULIANO