Endomorphin-1 analogs containing α-methyl-β-amino acids exhibit potent analgesic activity after peripheral administration

Y Wang, J Yang, X Liu, L Zhao, D Yang… - Organic & …, 2017 - pubs.rsc.org
This study describes the design and synthesis of endomorphin-1 analogs containing C-
terminal aromatic α-methyl-β-amino acids and an N-terminal native tyrosine or 2, 6-dimethyl …

[PDF][PDF] A Brief Survey on Recent Endomorphin-1 and Endomorphin-2 Analogues

R De Marco - J Biochem Chem Sci, 2017 - researchgate.net
The neurophysiological distribution of the Endomorphins (EMs), ie, Endomorphin-1 (EM1)
and Endomorphin-2 (EM2), reflects their potential role in many major biological processes …