The application of traditional medicine by humans for the treatment of ailments as well as
improving the quality of life far outdates recorded history. To date, a significant percentage of …

A highly enantioselective aza-Friedel–Crafts reaction of tryptanthrin-derived ketimines with
indoles/pyrrole using chiral phosphoric acid as a catalyst has been established. This …

A novel transition metal-free strategy for the synthesis of benzene-fused β-carboline
scaffolds has been developed. This protocol offers a rapid and direct pathway to access the …

Highly enantioselective access to tetrahydroxanthone compounds was achieved through
copper-bis (oxazoline)-catalyzed [4+ 2] cycloaddition of chrom-4-one dienophiles and …

We present a novel nickel-catalyzed reaction of indole-tethered 2-alkynylphenol esters with
various (hetero) aryl boronic acids, resulting in the synthesis of diversely functionalized …

The development of new anti-cancer agents is an urgent necessity nowadays, as it is one of
the major causes of mortality worldwide. Many drugs currently used are derived from natural …

We have developed a diversity‐oriented, substrate‐controlled, chemoselective synthetic
method for a variety of structurally diverse 1‐sulfonylquinazoline‐2, 4 (1H, 3H)‐diones and 2 …

A total synthesis of kopsone was achieved, featuring stereoselective preparation of an
acyclic aldehyde having a protected hydroxylamine moiety via Ireland–Claisen …

Dangkwisoo-san (DS) is a traditional Korean herbal medicine used to treat traumatic
diseases, including pulmonary contusions, traumatic pneumothorax, bruising, and ankle …

We present the preparation of a series of novel natural product‐like homobarrelenones,
norcaranes, and dihydrofluorenones through a diversity‐oriented synthetic (DOS) strategy …