Oral delivery of anticancer drugs: challenges and opportunities

K Thanki, RP Gangwal, AT Sangamwar… - Journal of controlled …, 2013 - Elsevier
The present report focuses on the various aspects of oral delivery of anticancer drugs. The
significance of oral delivery in cancer therapeutics has been highlighted which principally …

Recent advances in doxorubicin formulation to enhance pharmacokinetics and tumor targeting

J Lee, MK Choi, IS Song - Pharmaceuticals, 2023 - mdpi.com
Doxorubicin (DOX), a widely used drug in cancer chemotherapy, induces cell death via
multiple intracellular interactions, generating reactive oxygen species and DNA-adducted …

Co-encapsulation of tamoxifen and quercetin in polymeric nanoparticles: implications on oral bioavailability, antitumor efficacy, and drug-induced toxicity

AK Jain, K Thanki, S Jain - Molecular pharmaceutics, 2013 - ACS Publications
The present investigation reports the preparation, optimization, and characterization of orally
administrable PLGA-NPs co-encapsulated with tamoxifen (Tmx) and quercetin (QT). The …

Recent advances in drug delivery nanocarriers incorporated in temperature-sensitive Pluronic F-127–A critical review

RJ PJ, OS Oluwafemi, S Thomas, AO Oyedeji - Journal of Drug Delivery …, 2022 - Elsevier
New polymeric systems are constantly developed for novel biomedical applications.
Pluronic F127 (PF127) is a tri-block copolymer with surface-active properties. It comprises a …

HSA coated iron oxide nanoparticles as drug delivery vehicles for cancer therapy

Q Quan, J Xie, H Gao, M Yang, F Zhang… - Molecular …, 2011 - ACS Publications
An ongoing effort in the field of nanomedicine is to develop nanoplatforms with both imaging
and therapeutic functions, the “nanotheranostics”. We have previously developed a human …

Targeted therapy of breast tumor by PLGA-based nanostructures: The versatile function in doxorubicin delivery

TS Dongsar, TT Dongsar, N Molugulu… - Environmental …, 2023 - Elsevier
Breast carcinoma is a molecularly diverse illness, and it is among the most prominent and
often reported malignancies in female across the globe. Surgical intervention …

Nanostructured lipid carriers for oral bioavailability enhancement of exemestane: formulation design, in vitro, ex vivo, and in vivo studies

A Singh, YR Neupane, B Mangla, K Kohli - Journal of pharmaceutical …, 2019 - Elsevier
Exemestane (EXE) is a novel oral steroidal aromatase inhibitor approved for the treatment of
breast cancer. However, its oral clinical application is limited because of low aqueous …

Improved stability and antidiabetic potential of insulin containing folic acid functionalized polymer stabilized multilayered liposomes following oral administration

AK Agrawal, H Harde, K Thanki, S Jain - Biomacromolecules, 2014 - ACS Publications
The present study reports the folic acid (FA) functionalized insulin loaded stable liposomes
with improved bioavailability following oral administration. Liposomes were stabilized by …

Folate-decorated PLGA nanoparticles as a rationally designed vehicle for the oral delivery of insulin

S Jain, VV Rathi, AK Jain, M Das, C Godugu - Nanomedicine, 2012 - Taylor & Francis
Aims: The present study reports a novel approach for enhancing the oral absorption and
hypoglycemic activity of insulin via encapsulation in folate-(FA) coupled polyethylene glycol …

Terminal modification of polymeric micelles with π-conjugated moieties for efficient anticancer drug delivery

Y Liang, X Deng, L Zhang, X Peng, W Gao, J Cao, Z Gu… - Biomaterials, 2015 - Elsevier
High drug loading content is the critical factor to polymeric micelles for efficient
chemotherapy. Small molecules of cinnamic acid, 7-carboxymethoxy coumarin and chrysin …