Enhancing the solubility and bioactivity of anticancer drug tamoxifen by water-soluble pillar [6] arene-based host–guest complexation
Enhancing the solubility and bioactivity of anticancer drug tamoxifen by water-soluble pillar[6]arene-based
host–guest complexation - Chemical Communications (RSC Publishing) DOI:10.1039/C7CC05305C …
host–guest complexation - Chemical Communications (RSC Publishing) DOI:10.1039/C7CC05305C …
Oral bioavailability enhancement of raloxifene by developing microemulsion using D-optimal mixture design: optimization and in-vivo pharmacokinetic study
The objective of this work was to utilize a potential of microemulsion for the improvement in
oral bioavailability of raloxifene hydrochloride, a BCS class-II drug with 2% bioavailability …
oral bioavailability of raloxifene hydrochloride, a BCS class-II drug with 2% bioavailability …
Solubility determination of raloxifene hydrochloride in ten pure solvents at various temperatures: Thermodynamics-based analysis and solute–solvent interactions
The purpose of the present study was to determine the solubility of raloxifene hydrochloride
(RHCl) in ten solvents: water, ethanol, isopropyl alcohol (IPA), ethylene glycol (EG) …
(RHCl) in ten solvents: water, ethanol, isopropyl alcohol (IPA), ethylene glycol (EG) …
[PDF][PDF] Development of Risedronate Sodium-loaded Nanosponges by Experimental Design: Optimization and in vitro Characterization.
The present investigation focussed on the development of a novel strategy to enhance the
bioavailability of risedronate sodium, which has poor and erratic absorption. Nanosponges …
bioavailability of risedronate sodium, which has poor and erratic absorption. Nanosponges …
Poly (methyl vinyl ether-co-maleic acid) for enhancement of solubility, oral bioavailability and anti-osteoporotic effects of raloxifene hydrochloride
Raloxifene HCl (RH) has poor water solubility and due to its extensive first pass metabolism;
its bioavailability is only 2%. The purpose of the present study was to enhance the aqueous …
its bioavailability is only 2%. The purpose of the present study was to enhance the aqueous …
Formulation and characterization of raloxifene nanostructured lipid carriers for permeability and uptake enhancement applications
A Sharma, J Streets, P Bhatt, P Patel… - ASSAY and Drug …, 2022 - liebertpub.com
Raloxifene (RLX), a biopharmaceutical classification system (BCS) class II drug, is a
selective estrogen receptor modulator (SERM) having an estrogenic effect on the bone and …
selective estrogen receptor modulator (SERM) having an estrogenic effect on the bone and …
Study on protolytic equilibria and the effects of pH, cyclodextrins and polysorbate 80 on solubility of raloxifene hydrochloride
MR Popović-Nikolić, M Čakar, N Todorović, K Nikolić… - Chemical Papers, 2024 - Springer
The acid–base equilibria of raloxifene and the mutual influence of pH and solubility
enhancers on the solubility of raloxifene hydrochloride were studied. The apparent …
enhancers on the solubility of raloxifene hydrochloride were studied. The apparent …
Enhancement in dissolution profile of cilnidipine by nanonization technique: Optimization by box-behnken design
Objectives Cilnidipine has limited 25-30% of bioavailability due to BCS class II category
drug. The aim of present work was to improve the solubility followed by dissolution rate of …
drug. The aim of present work was to improve the solubility followed by dissolution rate of …
[PDF][PDF] Solubility and Dissolution Rate Enhancement of Poorly Soluble Telmisartan using Hydrotropy Method
N Shah - Asian Journal of Pharmaceutics (AJP), 2024 - asiapharmaceutics.info
Solubility and Dissolution Rate Enhancement of Poorly Soluble Telmisartan using Hydrotropy
Method Page 1 Asian Journal of Pharmaceutics • Jan-Mar 2024 • 18 (1) | 154 Solubility and …
Method Page 1 Asian Journal of Pharmaceutics • Jan-Mar 2024 • 18 (1) | 154 Solubility and …
[PDF][PDF] Luliconazole Loaded Niosomal Topical Gel: Factorial Design, in vitro Characterization and Antifungal Study
N Shah, R Prajapati, D Gohil… - Ind. J. Pharm …, 2023 - pdfs.semanticscholar.org
ABSTRACT Aim/Background: This research work intended to make use of prospective
advantages of niosomes for the improvement in topical delivery of poorly soluble …
advantages of niosomes for the improvement in topical delivery of poorly soluble …