[HTML][HTML] Cardiovascular activity

HG Vogel - Drug Discovery and Evaluation, 2008 - ncbi.nlm.nih.gov
PURPOSE AND RATIONALE α1-adrenoceptors are widely distributed and are activated
either by norepinephrine released from sympathetic nerve terminals or by epinephrine …

Cardiovascular Effects of LAS 30538, a New Vascular Selective Ca2+‐Channel Blocker

I Cardelus, J Bou, J Llenas, P Berga… - Journal of pharmacy …, 1992 - Wiley Online Library
A new compound, 1‐[2‐(2, 6‐dimethylphenoxy) ethyl]‐α, α‐bis‐(p‐fluorphenyl)‐4‐piperidine
methanol (LAS 30538), was found to have potent vasodilator effects. Its vasorelaxant activity …

Effects of P5, a novel oxazolo(3,2‐a)pyridine derivative with a long‐acting antihypertensive activity, on different agonist‐mediated pressor responses in pithed rats

E Martin, MA Sevilla, A Moran… - Journal of Autonomic …, 2001 - Wiley Online Library
1 An oxazolo (3, 2‐a) pyridine derivative P5, described chemically as (±)‐ethyl‐7‐(3‐
nitrophenyl)‐5, 8a‐dimethyl‐6‐methoxycarbonyl‐2, 3, 8, 8a‐tetrahydro‐7H‐oxazolo [3, 2‐a] …

Ursolic acid derivatives

AEGE Amr, MA Al-Omar, AA Almehizia… - US Patent …, 2019 - Google Patents
US10343997B1 - Ursolic acid derivatives - Google Patents US10343997B1 - Ursolic acid
derivatives - Google Patents Ursolic acid derivatives Download PDF Info Publication …

Cardiovascular activity

HG Vogel, WH Vogel - Drug Discovery and Evaluation: Pharmacological …, 1997 - Springer
The α-adrenoreceptor population of plasma membranes from rat heart ventricles consists
only of the α 1-adrenoreceptor subtype. A constant concentration of the radioligand 3 H …