Synthesis and biological evaluation of some 1‐naphthol derivatives as antioxidants, acetylcholinesterase, and carbonic anhydrase inhibitors
M Erdoğan, L Polat Köse, S Eşsiz… - Archiv der …, 2021 - Wiley Online Library
A series of some naphthol derivatives 4a–f, 5a, f, 6a, and 7a, b (six novel ones: 4c, d, 5a, 6a,
7a, b) bearing F, Cl, Br, OMe, and dioxole substituents at different positions of the aromatic …
7a, b) bearing F, Cl, Br, OMe, and dioxole substituents at different positions of the aromatic …
New 4-methanesulfonyloxy benzohydrazide derivatives as potential antioxidant and carbonic anhydrase I and II inhibitors: synthesis, characterization, molecular …
As an archetypal molecule, hydrazides have a crucial vital role in numerous applications, so
hydrazide-related inhibitors, especially sulfur-enriched, are favored. In the present work, we …
hydrazide-related inhibitors, especially sulfur-enriched, are favored. In the present work, we …
Evaluation of cytotoxic potentials of some isoindole-1, 3-dione derivatives on HeLa, C6 and A549 cancer cell lines
A Tan, AS Yaglioglu, NH Kishali, E Sahin… - Medicinal …, 2020 - ingentaconnect.com
Background: Norcantharimides are known as norcantharidine derivatives and contain an
isoindole skeleton structure. Isoindole derivatives have positive effect on inflammatory …
isoindole skeleton structure. Isoindole derivatives have positive effect on inflammatory …
Novel hybrid isoindole‐1,3(2H)‐dione compounds containing a 1H‐tetrazole moiety: Synthesis, biological evaluation, and molecular docking studies
In this study, novel hybrid isoindole‐1, 3 (2H)‐dione compounds (10 and 11) carrying a 1H‐
tetrazole moiety were synthesized, characterized and their inhibitory properties against …
tetrazole moiety were synthesized, characterized and their inhibitory properties against …
Dual delivery of platelet‐derived growth factor and bone morphogenetic factor‐6 on titanium surface to enhance the early period of implant osseointegration
Objective To test the surface properties and in vitro effects of a new sequential release
system on MC3T3‐E1 cells for improved osseointegration. Background BMP6‐loaded …
system on MC3T3‐E1 cells for improved osseointegration. Background BMP6‐loaded …
Synthesis, cytotoxicity, and antibacterial studies of 2,4,5,6‐substituted hexahydro‐1H‐isoindole‐1,3(2H)‐dione
E Yetişkin, Ö Gündoğdu, D Mete… - Chemical Biology & …, 2023 - Wiley Online Library
In this study, synthesis of novel isoindole‐1, 3‐dione analogues bearig halo, hydroxy, and
acetoxy groups at the position 4, 5, 6 of the bicyclic imide ring was performed to examine …
acetoxy groups at the position 4, 5, 6 of the bicyclic imide ring was performed to examine …
Evaluation of isoindole derivatives: Antioxidant potential and cytotoxicity in the HT‐29 colon cancer cells
A Kılıç Süloğlu, G Selmanoglu… - Archiv der …, 2020 - Wiley Online Library
Norcantharimides have an isoindole skeleton structure, and some isoindoline derivatives
have positive effects on inflammatory pathologies, including cancers. The present study …
have positive effects on inflammatory pathologies, including cancers. The present study …
Remarkable reactivity of boron-substituted furans in the Diels–Alder reactions with maleic anhydride
NS Medrán, F Dezotti, SC Pellegrinet - Organic letters, 2019 - ACS Publications
The reactivity of boron-substituted furans as dienes in the Diels–Alder reaction with maleic
anhydride has been investigated. Gratifyingly, the furans with boryl substituents at C-3 gave …
anhydride has been investigated. Gratifyingly, the furans with boryl substituents at C-3 gave …
Regio-and stereo-chemical ring-opening reactions of the 2, 3-epoxy alcohol derivative with nucleophiles: Explanation of the structures and C-2 selectivity supported …
The ring-opening reactions of (1aS, 2S, 6bR)-5-ethyl-2-hydroxyhexahydro-4H-oxireno [2, 3-
e] isoindole-4, 6 (5H)-dione were investigated under very mild and nonchelated conditions …
e] isoindole-4, 6 (5H)-dione were investigated under very mild and nonchelated conditions …
Synthesis and biological evaluation of new chloro/acetoxy substituted isoindole analogues as new tyrosine kinase inhibitors
We have developed a versatile synthetic approach for the synthesis of new isoindole
derivatives via the cleavage of ethers from tricyclic imide skeleton compounds. An exo …
derivatives via the cleavage of ethers from tricyclic imide skeleton compounds. An exo …