Recent years have seen a marked increase in the occurrence of sulfoximines in the
chemical sciences, often presented as valuable motifs for medicinal chemistry. This has …

Sulfur can form diverse S (IV) and S (VI) stereogenic centers, of which some have gained
significant attention recently due to their increasing use as pharmacophores in drug …

Achiral sulfur functional groups, such as sulfonamide, sulfone, thiol and thioether, are
common in drugs and natural products. By contrast, chiral sulfur functional groups are often …

Sulfoximines are widely used as medicines, agricultural chemicals, chiral precursors, and
chiral ligands in asymmetric synthesis, as well as pivotal intermediates for the construction of …

Sulfoximines and sulfonimidamides are promising compounds for medicinal and
agrochemistry. As monoaza analogues of sulfones and sulfonamides, respectively, they …

Chiral sulfimides, the aza‐analogues of sulfoxides, are valuable compounds in organic
synthesis and medicinal chemistry. Herein, we report an efficient method for preparing chiral …

Sulfonimidoyl halides have previously shown poor stability and selectivity in reaction with
organometallic reagents. Here we report the preparation of enantioenriched sulfonimidoyl …

A novel copper-catalyzed cross-coupling reaction of sulfinamides and aryl boronic acids is
developed. The reaction is highly chemoselective and stereospecific, which allows mild …

With unique chemical and biological activity, sulfoximines have attracted enormous attention
in the past decades, whereas limited reports exist for their synthesis via asymmetric …

The development of NH transfer reactions using hypervalent iodine and simple sources of
ammonia has facilitated the synthesis of sulfoximines and sulfonimidamides for applications …