The involvement of 1, 3-dipolar cycloaddition (1, 3-DP), double bond migration, metathesis,
and nitrile oxide (including in situ-generated nitrile oxide) as dipoles, together with the C= C …

Although there is an abundance of methods for the enantioselective synthesis of 2‐
isoxazolines and 2‐isoxazolin‐5‐ones, relatively few of these approaches have been …

Gold catalysis is an important method for alkyne functionalization. Here we report the gold‐
catalyzed formal [3+ 2] aminative cyclization of yndiamides and isoxazoles in a direct …

Acylation of nitroalkylmalonates was found to yield substituted isoxazoline derivatives. This
redox‐neutral transformation has a wide substrate scope and produces target products with …

A series of indolyl or imidazo [1, 2-a] pyridinyl-substituted para-quinone methides (p-QMs) is
prepared by a metal-free, TEMPO-mediated cross-dehydrogenative coupling of butylated …

An efficient [2+ 2+ 1] cycloaddition reaction of alkyl trifluorodiazoethane with nitrosoarenes
and alkynes has been described. This reaction is conducted under mild conditions with CuI …

Abstract The [3+ 2] cycloaddition reactions (32CA) between N-benzyl fluoro nitrone and
electron-deficient dipolarophiles alkynes have been studied using molecular electron …

An efficient K 2 CO 3-mediated intramolecular oxa-Michael cyclization of β, β-diarylated α, β-
unsaturated ketoximes is described. This methodology allows access to arene-rich 2 …

Yndiamides, doubly nitrogen-substituted alkynes, could serve as versatile precursors to
various 1, 2-diaminated products. This thesis focused on the gold-catalysed …

The isoxazoline ring has been utilized in many therapeutic agents. For example, it is the key
structure in ISO-1, an anti-inflammatory agent with unique anti-Type 1 diabetes activity …