[HTML][HTML] Successful oral delivery of poorly water-soluble drugs both depends on the intraluminal behavior of drugs and of appropriate advanced drug delivery systems

BJ Boyd, CAS Bergström, Z Vinarov, M Kuentz… - European Journal of …, 2019 - Elsevier
Poorly water-soluble drugs continue to be a problematic, yet important class of
pharmaceutical compounds for treatment of a wide range of diseases. Their prevalence in …

Self-nano-emulsifying drug-delivery systems: From the development to the current applications and challenges in oral drug delivery

AB Buya, A Beloqui, PB Memvanga, V Préat - Pharmaceutics, 2020 - mdpi.com
Approximately one third of newly discovered drug molecules show insufficient water
solubility and therefore low oral bio-availability. Self-nano-emulsifying drug-delivery systems …

INFOGEST static in vitro simulation of gastrointestinal food digestion

A Brodkorb, L Egger, M Alminger, P Alvito… - Nature protocols, 2019 - nature.com
Developing a mechanistic understanding of the impact of food structure and composition on
human health has increasingly involved simulating digestion in the upper gastrointestinal …

50 years of oral lipid-based formulations: provenance, progress and future perspectives

OM Feeney, MF Crum, CL McEvoy, NL Trevaskis… - Advanced drug delivery …, 2016 - Elsevier
Lipid based formulations (LBF) provide well proven opportunities to enhance the oral
absorption of drugs and drug candidates that sit close to, or beyond, the boundaries of …

Solid self emulsifying drug delivery system: Superior mode for oral delivery of hydrophobic cargos

I Maji, S Mahajan, A Sriram, P Medtiya… - Journal of Controlled …, 2021 - Elsevier
A significant proportion of recently approved drug molecules possess poor aqueous
solubility which further restrains their desired bioavailability. Poor aqueous solubility of these …

Effect of processing technologies on the digestibility of egg proteins

ZF Bhat, JD Morton, AEDA Bekhit… - … Reviews in Food …, 2021 - Wiley Online Library
Egg and egg products are a rich source of highly bioavailable animal proteins. Several
processing technologies can affect the structural and functional properties of these proteins …

In vitro digestion models to evaluate lipid based drug delivery systems; present status and current trends

R Berthelsen, M Klitgaard, T Rades… - Advanced Drug Delivery …, 2019 - Elsevier
During the past two decades, a range of in vitro models simulating the digestion processes
occurring in the stomach and small intestine have been developed to characterize lipid …

[HTML][HTML] Synergistic stabilization of emulsion gel by nanoparticles and surfactant enables 3D printing of lipid-rich solid oral dosage forms

J Johannesson, MM Pathare, M Johansson… - Journal of Colloid and …, 2023 - Elsevier
Pharmaceutical formulation of oral dosage forms is continuously challenged by the low
solubility of new drug candidates. Pickering emulsions, emulsions stabilized with solid …

[HTML][HTML] In vitro and in vivo correlation for lipid-based formulations: Current status and future perspectives

Y Huang, Q Yu, Z Chen, W Wu, Q Zhu, Y Lu - Acta Pharmaceutica Sinica B, 2021 - Elsevier
Lipid-based formulations (LBFs) have demonstrated a great potential in enhancing the oral
absorption of poorly water-soluble drugs. However, construction of in vitro and in vivo …

A proof of concept for 3D printing of solid lipid-based formulations of poorly water-soluble drugs to control formulation dispersion kinetics

K Vithani, A Goyanes, V Jannin, AW Basit… - Pharmaceutical …, 2019 - Springer
Purpose The use of three-dimensional printing (3DP) in the development of pharmaceutical
dosage forms is growing rapidly. However, the research is almost exclusively focussed on …