Novel promising benzoxazole/benzothiazole‐derived immunomodulatory agents: Design, synthesis, anticancer evaluation, and in silico ADMET analysis
Eleven novel benzoxazole/benzothiazole‐based thalidomide analogs were designed and
synthesized to obtain new effective antitumor immunomodulatory agents. The synthesized …
synthesized to obtain new effective antitumor immunomodulatory agents. The synthesized …
Synthesis of acridine cyclic imide hybrid molecules and their evaluation for anticancer activity
Amino acridine derivatives (1a–e) on condensation with dihydrofuran-2, 5-dione,
hexahydroisobenzofuran-1, 3-dione and isochroman-1, 3-dione under microwave irradiation …
hexahydroisobenzofuran-1, 3-dione and isochroman-1, 3-dione under microwave irradiation …
Synthesis, hypolipidemic, and anti-inflammatory activities of arylphthalimides
SPO Assis, TG Araújo, VLM Sena… - Medicinal Chemistry …, 2014 - Springer
Phthalimide and some N-substituted cyclic imides may be potent hypolipidemic agents,
capable of reducing plasma cholesterol, and triglyceride levels. In this work, N …
capable of reducing plasma cholesterol, and triglyceride levels. In this work, N …
Synthesis of N‐aminophalimides derived from α‐amino acids: Theoretical study to find them as HDAC8 inhibitors by docking simulations and in vitro assays
JE Guzmán Ramírez… - Chemical Biology & …, 2023 - Wiley Online Library
Phthalimides are valuable for synthesis and biological properties. New acetamides 3 (a–c)
and 4 (a–c) were synthesized and characterized as precursors for novel N‐aminophalimides …
and 4 (a–c) were synthesized and characterized as precursors for novel N‐aminophalimides …
Palladium-Catalyzed sp3 C–H Acetoxylation of α,α-Disubstituted α-Amino Acids
A Matsumura, Y Usuki, T Satoh - Chemistry, 2023 - mdpi.com
The sp3 C–H acetoxylation at the β-position of α, α-disubstituted α-amino acids proceeds
smoothly under palladium catalysis in the presence of PhI (OAc) 2. This reaction provides a …
smoothly under palladium catalysis in the presence of PhI (OAc) 2. This reaction provides a …
Solvent free, catalyst free, microwave or grinding assisted synthesis of bis-cyclic imide derivatives and their evaluation for anticancer activity
Cyclic imides are well known to be very important antitumor agents such as mitonafide and
amonafide etc. Based on this fact, we have synthesized two series of cyclic imide derivatives …
amonafide etc. Based on this fact, we have synthesized two series of cyclic imide derivatives …
Diphenic acid derivatives: Synthesis, reactions, and applications
MA Salem, MH Helel, YA Ammar… - Synthetic …, 2017 - Taylor & Francis
Full article: Diphenic acid derivatives: Synthesis, reactions, and applications Skip to Main
Content Taylor and Francis Online homepage Taylor and Francis Online homepage Log in …
Content Taylor and Francis Online homepage Taylor and Francis Online homepage Log in …
Design, Synthesis, Spectral Analysis and Molecular Docking Studies of Some Cyclic Imide as Potential Anti Breast and Cervical Cancer Agents
MAR Essa, AM Dhumad - International journal of health sciences - neliti.com
Design, synthesis, spectral analysis and molecular docking studies of some cyclic imide as
potential anti breast and cervical ca Page 1 How to Cite: Essa, MAR, & Dhumad, AM (2022) …
potential anti breast and cervical ca Page 1 How to Cite: Essa, MAR, & Dhumad, AM (2022) …
A multivariate statistical analysis of the QSAR of 2-(substituted phenyl) indan-1, 3-diones with hypolipidemic activity
AG Silva, MN Ramos - Journal of the Brazilian Chemical Society, 2012 - SciELO Brasil
Electronic descriptors obtained from AM1 molecular orbital calculations were employed,
along with the empirical parameters log P and π, in a multivariate statistical analysis of the …
along with the empirical parameters log P and π, in a multivariate statistical analysis of the …
[PDF][PDF] A multivariate statistical analysis of the quantitative structure-activity relationships (QSAR) of 2-(substituted phenyl) indan-1, 3-diones with hypolipidemic activity
AG da Silva, MN Ramosb - J. Braz. Chem. Soc, 2012 - SciELO Brasil
Electronic descriptors obtained from AM1 molecular orbital calculations were employed,
along with the empirical parameters log P and π, in a multivariate statistical analysis of the …
along with the empirical parameters log P and π, in a multivariate statistical analysis of the …