Advances in pyranopyrazole scaffolds' syntheses using sustainable catalysts—a review
Heterogeneous catalysis plays a crucial role in many chemical processes, including
advanced organic preparations and the design and synthesis of new organic moieties …
advanced organic preparations and the design and synthesis of new organic moieties …
[PDF][PDF] Synthesis, characterization and evaluation of some Pyranopyrazole derivatives as multifunction additives for medium lubricating Oils
AR Salih, ZAK Al-Messri - Iraqi Journal of Science, 2022 - iasj.net
The current work involves synthesis of 6-amino-4-(4-hydroxyl-3-methoxyphenyl)-3-methyl-1-
phenyl-1, 4- dihydropyrano [2, 3-c] pyrazole-5-carbonitrile (2) by condensation of 2-(4 …
phenyl-1, 4- dihydropyrano [2, 3-c] pyrazole-5-carbonitrile (2) by condensation of 2-(4 …
Visible-light induced acridinium catalysed synthesis of biologically active dihydropyranopyrazoles scaffolds via HAT
Visible light driven acridinium catalysed synthesis of dihydropyranopyrazole scaffolds from
pyrazol and butyne derivatives under an air atmosphere is reported at room temperature …
pyrazol and butyne derivatives under an air atmosphere is reported at room temperature …
Molecular modelling, synthesis and antimicrobial evaluation of benzimidazole nucleoside mimetics
H Chaurasia, VK Singh, R Mishra, AK Yadav… - Bioorganic …, 2021 - Elsevier
A series of new N-1-(β-d-ribofuranosyl) benzimidazole derivatives has been designed using
in silico methods and synthesized as probable antimicrobial agents. Further, the compounds …
in silico methods and synthesized as probable antimicrobial agents. Further, the compounds …
Targeting disease with benzoxazoles: a comprehensive review of recent developments
A Abdullahi, KY Yeong - Medicinal Chemistry Research, 2024 - Springer
Benzoxazole is an attractive scaffold in medicinal chemistry due to its diverse biological
applications. From 2016 to 2023, a plethora of benzoxazole derivatives have been …
applications. From 2016 to 2023, a plethora of benzoxazole derivatives have been …
2-Aminobenzoxazole-appended coumarins as potent and selective inhibitors of tumour-associated carbonic anhydrases
A Fuentes-Aguilar, P Merino-Montiel… - Journal of Enzyme …, 2022 - Taylor & Francis
We have carried out the design, synthesis, and evaluation of a small library of 2-
aminobenzoxazole-appended coumarins as novel inhibitors of tumour-related CAs IX and …
aminobenzoxazole-appended coumarins as novel inhibitors of tumour-related CAs IX and …
Design, docking, molecular dynamics, synthesis and antimicrobial studies on quinoline derivatives and some isosteres
The computer added design, synthesis, antibacterial and antifungal activities of a series of
quinoline derivatives and some isosteres are reported. In silico studies using autodock …
quinoline derivatives and some isosteres are reported. In silico studies using autodock …
Introducing of novel class of pyrano[2,3-c]pyrazole-5-carbonitrile analogs with potent antimicrobial activity, DNA gyrase inhibition, and prominent pharmacokinetic …
Microbiological DNA gyrase is recognized as an exceptional microbial target for the
innovative development of low-resistant and more effective antimicrobial drugs. Hence, we …
innovative development of low-resistant and more effective antimicrobial drugs. Hence, we …
Molecular docking and antibacterial studies of pyranopyrazole derivatives synthesized using [Pap-Glu@ Chi] biocatalyst through a greener approach
In the present work, papain enzyme was immobilized on a polymer support chitosan through
a linkage of glutaraldehyde to form the [Pap-Glu@ Chi] biocatalyst through the covalent …
a linkage of glutaraldehyde to form the [Pap-Glu@ Chi] biocatalyst through the covalent …
Synthesis and characterization of derivatives including thiazolidine-2,4-dione/1-H- imidazole and evaluation of antimicrobial, antioxidant, and cytotoxic properties of …
HY Nyaki, NO Mahmoodi - Research on Chemical Intermediates, 2021 - Springer
Several new derivatives of thiazolidine-2, 4-dione and 1-H-imidazole were prepared using
imidazole aldehydes 6a–6f in ethanol as a solvent. Products 7a–7f were obtained in …
imidazole aldehydes 6a–6f in ethanol as a solvent. Products 7a–7f were obtained in …