In vivo deposition of poorly soluble drugs

Z Lou, C Mu, CD Corpstein, T Li - Advanced Drug Delivery Reviews, 2024 - Elsevier
Administered drug molecules, whether dissolved or solubilized, have the potential to
precipitate and accumulate as solid forms in tissues and cells within the body. This phase …

[HTML][HTML] Therapeutic efficiency of Tamoxifen/Orlistat nanocrystals against solid ehrlich carcinoma via targeting TXNIP/HIF1-α/MMP-9/P27 and BAX/Bcl2/P53 signaling …

TA El-Masry, MMF El-Nagar, GA Oriquat… - Biomedicine & …, 2024 - Elsevier
Abstract Background Orlistat (Orli) is an anti-obesity medication that has been approved by
the US Food and Drug Administration. It has relatively limited oral bioavailability with …

[HTML][HTML] Anticancer Effect of Cycas media: Molecular Basis Through Modulation of PI3K/AKT/mTOR Signaling Pathway

J Alqahtani, EM Mosalam, HE Abo Mansour, AI Elberri… - Molecules, 2024 - mdpi.com
Many researchers are focusing on screening the biological activities of plants owing to their
safety and possible pharmacological actions. Consequently, we aimed to explore the …

Dioon rzedowskii: An antioxidant, antibacterial and anticancer plant extract with multi-faceted effects on cell growth and molecular signaling

WA Negm, E Elekhnawy, S Mahgoub… - International …, 2024 - Elsevier
This study investigated the antioxidant, anticancer, antibacterial properties of Dioon
rzedowskii extract, which had not been previously explored. We aimed to determine the …

[HTML][HTML] Potential Protective Effect of Orlistat: A Formulation of Nanocrystals Targeting Inflammation, Oxidative Stress, and Apoptosis in an Experimental Model of …

M Alsunbul, TA El-Masry, EI El Zahaby, MMS Gaballa… - Pharmaceutics, 2024 - mdpi.com
Background: Doxorubicin (DOX) is a widely used chemotherapeutic agent; nevertheless,
cardiotoxicity limits its effectiveness. Orlistat (Orli) is an irreversible lipase enzyme inhibitor …