Synthesis and biological evaluation of novel oxadiazole derivatives: A new class of thymidine phosphorylase inhibitors as potential anti-tumor agents

SA Shahzad, M Yar, M Bajda, B Jadoon… - Bioorganic & medicinal …, 2014 - Elsevier
Based on the fact that the thymidine phosphorylase inhibitors are considered potential anti-
tumor agents, a range of novel oxadiazole derivatives 3a–3u was designed and synthesized …

Efficient oxidative cyclization of N-acylhydrazones for the synthesis of 2,5-disubstituted 1,3,4-oxadiazoles using t-BuOI under neutral conditions

P Gao, Y Wei - Heterocyclic Communications, 2013 - degruyter.com
An efficient procedure for the oxidative cyclization of N-acylhydrazones was developed
utilizing tert-butyl hypoiodite (t-BuOI), which is generated in situ from t-BuOCl and NaI. A …

Schiff bases of 3-formylchromones as antibacterial, antifungal, and phytotoxic agents (Supplementry Table)

KM Khan, A Ahmad, N Ambreen… - Letters in Drug …, 2009 - ingentaconnect.com
3-Formylchromone (1), 3-methyl-7-hydroxychromone (2) and Schiff Bases of 3-
formylchromone 3-25 have been synthesized and their antibacterial, antifungal and …

Effective end group modification of poly (3-hexylthiophene) with functional electron-deficient moieties for performance improvement in polymer solar cell

CM Chen, TH Jen, SA Chen - ACS applied materials & interfaces, 2015 - ACS Publications
A series of end-functionalized poly (3-hexylthiophene) s (P3HTs) were synthesized by end-
capping with electron-deficient moieties (EDMs, oxadiazole (OXD) and triazole (TAZ)) to …

Synthesis and biological activity of 2-(4, 5-dihydroisoxazol-5-yl)-1, 3, 4-oxadiazoles

KA Milinkevich, CL Yoo, TC Sparks… - Bioorganic & medicinal …, 2009 - Elsevier
Acid hydrazides were coupled with acrylic acid derivatives and cyclodehydration gave 1, 3,
4-oxadiazoles. Lastly, in-situ nitrile oxide formation from aryl oximes treated with sodium …

Antibiofilm potential of synthetic 2-amino-5-chlorobenzophenone Schiff bases and its confirmation through fluorescence microscopy

AK Khan, KM Khan, A Ahmed, M Taha, S Perveen - Microbial …, 2017 - Elsevier
Antibacterial/antibiofilm potential of microwave-assisted synthetic thirty-three 2-amino-5-
chloro benzophenone Schiff bases have been carried out against four bacterial strains ie …

Syntheses and antibacterial activity of Schiff bases from 16-isopropyl-5, 9-dimethyltetracyclo [10.2.2.01, 10.04, 9] hexadec-15-ene-5, 14-dicarboxylic acid

J Li, J Song, SB Shang, XP Rao… - Natural Product …, 2013 - Taylor & Francis
16-Isopropyl-5, 9-dimethyltetracyclo [10.2. 2.01, 10.04, 9] hexadec-15-ene-5, 14-dicarboxylic
acid (1b) was prepared from rosin through a Diels–Alder addition reaction. Then, a group of …

3-Substituted isocoumarins as thymidine phosphorylase inhibitors

KM Khan, S Ahmed, S Hussain, NA snm… - Letters in Drug …, 2010 - benthamdirect.com
3-Substituted isocoumarins 1-19 were synthesized and evaluated for their thymidine
phosphorylase inhibitory activity. Eight (8) compounds exhibited a varying degree of …

Synthesis, Antibacterial and Antifungal Activities of 3-Amino-5-methyl [1, 1'-biphenyl]-2, 4-dicarbonitrile Derivatives

K Mohammed Khan, W Jamil… - Letters in Drug …, 2012 - ingentaconnect.com
3-Amino-5-methyl-2, 4-dicarbonitrile biphenyl derivatives 1-14 have been synthesized and
all compounds were screened for their antibacterial effects against fourteen Gram-positive …

[PDF][PDF] Synthesis of new coumarin based acetohydrazones, their correspounding oxadiazoles and oxadiazolines, and the investigation of their antibacterial activity

N Baharvand, E Mottaghinejad… - Journal of Chemical …, 2023 - journals.iau.ir
Here we provide a report on the synthesis, structural recognition and tautomeric behavior of
a new series of coumarin-based hydrazide-hydrazones (4-methylcoumarin-7-yl-oxymethyl …