Regiodivergent Synthesis of 4‐and 5‐Sulfenyl Oxazoles from Alkynyl Thioethers

P Sekar, A Gupta, LE English… - … A European Journal, 2024 - Wiley Online Library
The regiodivergent synthesis of 4‐and 5‐sulfenyl oxazoles from 1, 4, 2‐dioxazoles and
alkynyl thioethers has been achieved. Gold‐catalysed conditions are used to favour the …

Photocatalytic Benzylic C–H Oxidation/Cyclization of Enaminones to the Synthesis of Polysubstituted Oxazoles

M Li, Z He, W Zhao, Y Yu, F Huang… - The Journal of Organic …, 2023 - ACS Publications
Photocatalytic benzylic C–H oxidation/cyclization of enaminones was efficiently achieved to
afford oxazole derivatives under mild conditions. The oxygen in the oxazole ring originated …

Deoxygenative Geminal Silylboration of Amides Using Silylboronates: Synthesis and Use of α‐Boryl‐α‐Silylalkylamines

K Watanabe, K Nagao, H Ohmiya - … Chemie International Edition, 2024 - Wiley Online Library
Abstract α‐Silylalkylamines and α‐borylalkylamines are versatile synthetic intermediates
and attractive scaffolds found in pharmaceutical drugs and agrochemicals. Despite great …

[PDF][PDF] Identification of diagnostic biomarkers and immuno-infiltration analysis for rheumatoid arthritis based on biological information and WGCNA.

Y Zhang, QY Yang, LS Yang, J Zhang… - European Review for …, 2023 - europeanreview.org
OBJECTIVE: Rheumatoid arthritis (RA), as an autoimmune disease, poses a huge social
and economic burden worldwide. Although the diagnosis of RA has been gradually …

[PDF][PDF] Development, characterization, and pharmacological investigation of sesamol and thymol conjugates of mefenamic acid

B Nija, A Rasheed, A Kottaimuthu - J. Evol. Med. Dent. Sci, 2020 - researchgate.net
BACKGROUND Prodrug technology was extensively employed in the drug discovery
processes and many approved drugs in the pharmaceutical industry were developed by the …

[PDF][PDF] Development, characterization and pharmacological investigation of umbelliferone conjugates of NSAIDs

B Nija, A Rasheed, A Kottaimuthu - … Sciences (P-ISSN 1683-3597 E-ISSN …, 2021 - iasj.net
The present investigation developed the ester prodrugs of Non-steroidal anti-inflammatory
drugs (NSAIDs), Mefenamic acid (MA) and Flurbiprofen (FBN) by conjugating with the …

奥沙普秦丹皮酚酯的合成及抗炎活性研究

徐学涛, 陈洁, 林芷晴, 李冬利, 张焜, 盛钊君, 王少华… - 有机化学, 2019 - sioc-journal.cn
有机化学 Page 1 有机化学 Chinese Journal of Organic Chemistry NOTE * Corresponding
authors. E-mail: wyuchemszj@126.com; wangshh@lzu.edu.cn Received March 12, 2019; …

Chromatographic profile, in silico and in vivo study of the pharmacokinetic and toxicological properties of major constituent present in kefir, the kefiran

SÉL Barros, HB de Lima, LKA Gonçalves… - Toxicology …, 2022 - academic.oup.com
Kefiran is a polysaccharide present in kefir grains that have been widely explored due to its
potential health benefits. The objective of this work was to characterize and quantify the …

Synthesis and Anti-inflammatory Effects of Oxaprozin-Paeonol Ester

X Xu, J Chen, Z Lin, D Li, K Zhang, Z Sheng… - Chinese Journal of …, 2019 - sioc-journal.cn
有机化学 Page 1 有机化学 Chinese Journal of Organic Chemistry NOTE * Corresponding
authors. E-mail: wyuchemszj@126.com; wangshh@lzu.edu.cn Received March 12, 2019; …