Mitochondria-targeting 1, 5-diazacyclooctane-spacered triterpene rhodamine conjugates exhibit cytotoxicity at sub-nanomolar concentration against breast cancer …
N Heise, S Becker, T Mueller, M Bache, R Csuk… - International Journal of …, 2023 - mdpi.com
1, 5-Diazacyclooctane was prepared by a simple synthetic sequence and coupled to
pentacyclic triterpenoic acids oleanolic acid, ursolic acid, betulinic acid, platanic acid, and …
pentacyclic triterpenoic acids oleanolic acid, ursolic acid, betulinic acid, platanic acid, and …
Supramolecular daisy chains
PR Ashton, I Baxter, SJ Cantrill… - Angewandte Chemie …, 1998 - Wiley Online Library
Our childhoods may be recalled when a self‐complementary cation, endowed with both a
dibenzo [24] crown‐8 macroring and a secondary dialkylammonium sidearm, self …
dibenzo [24] crown‐8 macroring and a secondary dialkylammonium sidearm, self …
Catenated cyclodextrins
D Armspach, PR Ashton, R Ballardini… - … A European Journal, 1995 - Wiley Online Library
A novel synthetic approach is described for the construction of catenanes in aqueous
solution from a partially methylated cyclodextrin (CD)‐namely, heptakis (2, 6‐di‐O‐methyl‐β …
solution from a partially methylated cyclodextrin (CD)‐namely, heptakis (2, 6‐di‐O‐methyl‐β …
Recognition of bipyridinium-based derivatives by hydroquinone-and/or dioxynaphthalene-based macrocyclic polyethers: From inclusion complexes to the self …
M Asakawa, PR Ashton, SE Boyd… - The Journal of …, 1997 - ACS Publications
A range of π-electron-rich macrocyclic polyethers incorporating dioxybenzene
(hydroquinone) and/or dioxynaphthalene units have been synthesized in good yields by …
(hydroquinone) and/or dioxynaphthalene units have been synthesized in good yields by …
A new design strategy for molecular recognition in heterogeneous systems: a universal crystal-face growth inhibitor for barium sulfate
PV Coveney, R Davey, JLW Griffin, Y He… - Journal of the …, 2000 - ACS Publications
Controlling crystallization in both chemical production and product formulations is well-
known. 1-4 As well as composition and temperature, specific additives can also exert a …
known. 1-4 As well as composition and temperature, specific additives can also exert a …
Developing an Amide-Spacered Triterpenoid Rhodamine Hybrid of Nano-Molar Cytotoxicity Combined with Excellent Tumor Cell/Non-Tumor Cell Selectivity
NV Heise, TC Denner, S Becker, S Hoenke, R Csuk - Molecules, 2023 - mdpi.com
Asiatic acid, a pentacyclic triterpene, was converted into a series of piperazinyl,
homopiperazinyl, and 1, 5-diazocinyl spacered rhodamine conjugates, differing in the type …
homopiperazinyl, and 1, 5-diazocinyl spacered rhodamine conjugates, differing in the type …
Copper (II) and zinc (II) complexation with N-ethylene hydroxycyclams and consequences on the macrocyclic backbone configuration
N AlHaddad, E Lelong, JM Suh, M Cordier… - Dalton …, 2022 - pubs.rsc.org
We report a series of four cyclams and cross-bridged cyclams, N-functionalized by one
hydroxyethyl arm, which may incorporate additional methyl (s) group (s). The Cu (II) and Zn …
hydroxyethyl arm, which may incorporate additional methyl (s) group (s). The Cu (II) and Zn …
Large-scale synthesis of the bifunctional chelating agent 2-(p-nitrobenzyl)-1, 4, 7, 10-tetraazacyclododecane-N, N', N'', N'''-tetraacetic acid, and the determination of its …
O Renn, CF Meares - Bioconjugate chemistry, 1992 - ACS Publications
The attachment of radiometals to monoclonal antibodies for medical applications requires
extreme stability under physiological conditions, with no significant release of metal …
extreme stability under physiological conditions, with no significant release of metal …
(π-Allyl)palladium Complexes with N,N'-Diphenylbispidinone Derivatives as a New Type of Chelating Nitrogen Ligand: Complexation Studies, Spectroscopic Properties, and …
A Gogoll, H Grennberg, A Axén - Organometallics, 1997 - ACS Publications
A series of 3, 7-diazabicyclo [3.3. 1] nonane (bispidine) derivatives have been synthesized,
and their properties as bidentate nitrogen ligands for (π-allyl) palladium complexes have …
and their properties as bidentate nitrogen ligands for (π-allyl) palladium complexes have …
Synthesis and conformational analysis of 2, 9-disubstituted 1-oxaquinolizidines
L Boerjesson, I Csoeregh, CJ Welch - The Journal of Organic …, 1995 - ACS Publications
The synthesis of (2S, 9JZ, 10S)-9-(5-(«erf-butyldiphenylsilyl) oxy) pentyl)-2-(hydroxymethyl)-l-
oxa-quinolizidine (29a) from (S)-malic acid, 1, 5-pentanediol, andtrifluoroacetamide is …
oxa-quinolizidine (29a) from (S)-malic acid, 1, 5-pentanediol, andtrifluoroacetamide is …