Quinoline hydrazide/hydrazone derivatives: Recent insights on antibacterial activity and mechanism of action

S Verma, S Lal, R Narang, K Sudhakar - ChemMedChem, 2023 - Wiley Online Library
Antibiotics are becoming gradually ineffective due to drug resistance, leading to greater
difficulty in the treatment of infectious diseases. Therefore, the development of new chemical …

Hypervalent‐Iodine (III)‐Mediated Oxidative Methodology for the Synthesis of Fused Triazoles

R Kamal, V Kumar, R Kumar - Chemistry–An Asian Journal, 2016 - Wiley Online Library
The organic chemistry of hypervalent organoiodine compounds has been an area of
unprecedented development. This surge in interest in the use of hypervalent iodine …

[PDF][PDF] Phytochemical and pharmacological properties of flavonols

A Sharma, P Sharma, HS Tuli, AK Sharma - eLS, 2018 - researchgate.net
Flavonoids are polyphenolic compounds, which are ubiquitous in nature and have been
categorised into flavonols, flavones, flavanones, isoflavones, catechins, anthocyanidins and …

Hantzsch‐like synthesis, DNA photocleavage, DNA/BSA binding, and molecular docking studies of bis (sulfanediyl) bis (tetrahydro‐5‐deazaflavin) analogs linked to …

MA Ragheb, RE Abdelwahab… - Chemistry & …, 2022 - Wiley Online Library
The cyclocondensation reaction of aldehydes with dimedone and bis (6‐aminopyrimidin‐4‐
one) in acetic acid led to the formation of the corresponding bis (pyrimido [4, 5‐b] quinoline …

Three Component One-Pot Synthesis and Antiproliferative Activity of New [1,2,4]Triazolo[4,3-a]pyrimidines

M Ben Hassen, D Msalbi, B Jismy, F Elghali, S Aifa… - Molecules, 2023 - mdpi.com
A series of new [1, 2, 4] triazolo [4, 3-a] pyrimidine derivatives was prepared using a one-pot
three-component synthesis from 5-amino-1-phenyl-1 H-1, 2, 4-triazoles, aromatic aldehydes …

Targeted potent antimicrobial benzochromene-based analogues: Synthesis, computational studies, and inhibitory effect against 14α-Demethylase and DNA Gyrase

AM Fouda, AH Hassan, EM Eliwa, HEA Ahmed… - Bioorganic …, 2020 - Elsevier
Abstract 7H-Benzo [7, 8] chromeno [2, 3-d] pyrimidin-9 (8H)-amine (6a, b) have been
synthesized via hydrazinolysis of the imidates (5a, b). Polysubstituted …

Synthesis, characterization, and antibacterial activity of some thiazoles derived from allyl thioureas

R Khare, J Sharma, A Sharma - Russian Journal of General Chemistry, 2016 - Springer
Synthesis of thiazoles was carried out from allyl thioureas using different cyclizing agents
such as hydrogen chloride gas and bromine. Synthesized compounds were characterized …

An effective and facile synthesis of new blue fluorophores on the basis of an 8-azapurine core

AK Eltyshev, PO Suntsova, KD Karmatskaia… - Organic & …, 2018 - pubs.rsc.org
A convenient synthesis of 2-aryl-2, 4-dihydro-5H-[1, 2, 3] triazolo [4, 5-d] pyrimidin-5-ones
(DTPs) from 3, 3-diamino-2-(arylazo) acrylonitriles through a versatile and readily accessible …

Chemistry and synthetic overview of flavonoids

A Sharma, H Singh Tuli, AK Sharma - … Aspects of Flavonoids: Their Role in …, 2019 - Springer
Flavonoids are widely distributed secondary metabolites in plants that are known to be
present in different vegetables and fruits. The flavonoid groups include various subclasses …

Flavones: Flavonoids having chemico-biological properties with a preview into anticancer action mechanism

A Sharma, HS Tuli, D Kashyap, AK Sharma - Bioactive Natural Products …, 2019 - Springer
Flavones belong to the flavonoids class of plant polyphenols. Owing to their widespread
distribution in plants, such as fruits, vegetables, herbs, spices, and beverages (tea, coffee …