Isoxazoles are important five‐membered aromatic heterocycles in organic chemistry.
Recently, many exciting advances in the synthesis and functionalization of isoxazoles have …

Modern organic synthesis requires easily obtainable chiral building blocks that show high
chemical versatility for their application in diverse synthetic processes. The main purpose of …

The results of the study on reactions of halogenoximes bearing (protected) functional groups
or fluorinated substituents with various phosphorus-containing dipolarophiles are described …

Abstract An efficient NaNO2/I2‐mediated one‐pot transformation of Morita–Baylis–Hillman
(MBH) acetates into alkyl 3‐nitro‐5‐(aryl/alkyl) isoxazole‐4‐carboxylates is described. In a …

Isoxazole derivatives are an important group of chemotherapeutic prototypes. In the current
study, we have synthesized few isoxazole derivatives and tested them for their …

Efficient routes for the regioselective synthesis of 3, 5‐bis (het) arylisoxazoles with
complementary regioselectivity have been developed. The methods involve the …

Nitro-substituted isoxazoles are of utmost interest both as versatile intermediates for targeted
organic synthesis and as perspective bioactive compounds for drug development …

The first example of the use of potassium trinitromethanide as a 1, 1-ambiphilic synthon
equivalent for the construction of a benzofuran moiety mediated by triethylamine has been …

A new approach to the synthesis of 3-nitroisoxazoles and 3-nitroisoxazolines based on the
[3+ 2]-cycloaddition of nitroformonitrile oxide (NFNO), generated by the cycloreversion of …

A new, selective method for the synthesis of (E)-vinyl sulfones is presence by palladium-
catalyzed C− S bond cleavage/conjugate addition. In the presence of Pd (OAc) 2 and …