The preparation methods and reactions of isoxazoles are described and systematized on
the basis of analysis of the literature published from 2005 to present. In the discussion of …

The need for precise and flexible synthetic methodology to underpin modern research in
chemical biology and materials science has fuelled a resurgence of interest in Huisgen 1, 3 …

Abstract Chloramine-T (CAT), the sodium salt of N-chloro-p-toluenesulfonamide, is a low-
cost mild oxidizing agent with a wide range of uses. Most importantly, it can be used in …

N-Protected amino acids can be easily converted into chiral α-amino aldehydes in a one-pot
reaction by activation with CDI followed by reduction with DIBAL-H. This method delivers …

A practical multigram metal free synthesis of isoxazole-containing building blocks from
commercially available amino acids was elaborated. The key reaction was a regioselective …

A tetrahydro-4 H-(pyrrolo [3, 4-d] isoxazol-3-yl) methanamine scaffold was designed as a
diamino derivative to stabilize parallel turn conformations. Its synthesis took advantage of a …

A convenient and efficient synthesis of novel achiral and chiral heterocyclic amino acid-like
building blocks was developed. Regioisomeric methyl 5-(N-Boc-cycloaminyl)-1, 2-oxazole-4 …

Here, we have reported an efficient one‐pot, three‐component reaction between various
aryl aldehydes, NH2OH. HCl, and propargyl alcohol using Ni‐Fe2O4 as a nanocatalyst …

Isoxazoles, isoxazolines and isoxazolidines are a class of heterocyclic compounds having a
remarkable number of applications and are very versatile building blocks in organic …

Изоксазолы проявляют широкий спектр биологической активности и демонстрируют
ряд необычных физико-химических свойств, в связи с чем находят применение в …