[HTML][HTML] Advances in computational structure-based antibody design

AM Hummer, B Abanades, CM Deane - Current opinion in structural biology, 2022 - Elsevier
Antibodies are currently the most important class of biotherapeutics and are used to treat
numerous diseases. Recent advances in computational methods are ushering in a new era …

Approaches to expand the conventional toolbox for discovery and selection of antibodies with drug-like physicochemical properties

HL Svilenov, P Arosio, T Menzen, P Tessier… - MAbs, 2023 - Taylor & Francis
Antibody drugs should exhibit not only high-binding affinity for their target antigens but also
favorable physicochemical drug-like properties. Such drug-like biophysical properties are …

Germline-encoded amino acid–binding motifs drive immunodominant public antibody responses

EL Shrock, RT Timms, T Kula, EL Mena, AP West Jr… - Science, 2023 - science.org
Despite the vast diversity of the antibody repertoire, infected individuals often mount
antibody responses to precisely the same epitopes within antigens. The immunological …

ImmuneBuilder: Deep-Learning models for predicting the structures of immune proteins

B Abanades, WK Wong, F Boyles, G Georges… - Communications …, 2023 - nature.com
Immune receptor proteins play a key role in the immune system and have shown great
promise as biotherapeutics. The structure of these proteins is critical for understanding their …

The 2022 Nucleic Acids Research database issue and the online molecular biology database collection

DJ Rigden, XM Fernández - Nucleic acids research, 2022 - academic.oup.com
Abstract The 2022 Nucleic Acids Research Database Issue contains 185 papers, including
87 papers reporting on new databases and 85 updates from resources previously published …

Toward real-world automated antibody design with combinatorial Bayesian optimization

A Khan, AI Cowen-Rivers, A Grosnit, PA Robert… - Cell Reports …, 2023 - cell.com
Antibodies are multimeric proteins capable of highly specific molecular recognition. The
complementarity determining region 3 of the antibody variable heavy chain (CDRH3) often …

Unsupervised protein-ligand binding energy prediction via neural euler's rotation equation

W Jin, S Sarkizova, X Chen… - Advances in Neural …, 2024 - proceedings.neurips.cc
Protein-ligand binding prediction is a fundamental problem in AI-driven drug discovery.
Previous work focused on supervised learning methods for small molecules where binding …

The Patent and Literature Antibody Database (PLAbDab): an evolving reference set of functionally diverse, literature-annotated antibody sequences and structures

B Abanades, TH Olsen, MIJ Raybould… - Nucleic Acids …, 2024 - academic.oup.com
Antibodies are key proteins of the adaptive immune system, and there exists a large body of
academic literature and patents dedicated to their study and concomitant conversion into …

A machine learning strategy for the identification of key in silico descriptors and prediction models for IgG monoclonal antibody developability properties

AB Waight, D Prihoda, R Shrestha, K Metcalf, M Bailly… - MAbs, 2023 - Taylor & Francis
Identification of favorable biophysical properties for protein therapeutics as part of
developability assessment is a crucial part of the preclinical development process …

Towards the accurate modelling of antibody− antigen complexes from sequence using machine learning and information-driven docking

M Giulini, C Schneider, D Cutting, N Desai… - …, 2024 - academic.oup.com
Motivation Antibody− antigen complex modelling is an important step in computational
workflows for therapeutic antibody design. While experimentally determined structures of …