Assessment of Anti-tyrosinase and Antioxidant Activities along with Molecular Docking Studies, and in silico ADME of Some 3-Hydroxypyridin-4-one Derivatives.
F Zare, S Sadeghian… - Trends in …, 2024 - search.ebscohost.com
Tyrosinase is an essential enzyme in melanin production, which plays an important role in
the browning of plants and vegetables and skin diseases in humans. Therefore, the design …
the browning of plants and vegetables and skin diseases in humans. Therefore, the design …
Structure Modification: Effect Of Lipophilic, Electronic, And Steric Parameters Of N-Benzoyln'-Phenylthiourea Compounds On Antiviral Activity Of Covid-19 By In Silico
N-benzoyl-N'-phenylthiourea (BFTU) compound is similar to amprenavir derivatives in the
urea compound, chloroquine in the-NH group, and the benzene ring, which is a potent …
urea compound, chloroquine in the-NH group, and the benzene ring, which is a potent …
Anticancer activity of N-(4-t-butylbenzoyl)-N'-phenylthiourea: Molecular docking, synthesis, and cytotoxic activity in breast and cervical cancer cells [Actividad …
D Kesuma, A Kirtishanti… - Journal of Pharmacy …, 2023 - repository.ubaya.ac.id
Context: N-(4-t-butylbenzoyl)-N'-phenylthiourea, a derivative compound of N-benzoyl-N'-
phenylthiourea, has relatively high lipophilicity with the epidermal growth factor receptor and …
phenylthiourea, has relatively high lipophilicity with the epidermal growth factor receptor and …
Molecular Docking And Biological Activity Of N-(4-Methoxy)-Benzoyl-N'-Phenylthiourea And N-(4-Trifluoro)-Benzoyl-N'-Phenylthiourea As Antibreast Cancer …
D Kesuma, S Siswandono… - Rasayan Journal of …, 2022 - repository.ubaya.ac.id
Current breast cancer therapy does not always work optimally, and cases of resistance have
been reported. Therefore, it is imperative to develop new effective drugs with minimal side …
been reported. Therefore, it is imperative to develop new effective drugs with minimal side …
THE POTENCY OF 4-NITROBENZOYL-3-ALLYLTHIOUREA AS AN AGENT OF BREAST CANCER WITH EGFR/HER2: IN SILICO AND IN VITRO STUDY.
T Widiandani, BT Purwanto - Rasayan Journal of …, 2022 - search.ebscohost.com
The objectives of this research were to predict the ADMET, docking, and investigate the
cytotoxicity activity of 4-nitrobenzoyl-3-allylthiourea (BATU-11) on MCF7 and MCF7/HER2 …
cytotoxicity activity of 4-nitrobenzoyl-3-allylthiourea (BATU-11) on MCF7 and MCF7/HER2 …
Thiourea Derivatives as Estrogen Receptor Alpha Inhibitors for Breast Cancer Therapy: An In Silico Evaluation with ADMET Prediction and Molecular Docking
H Puspaweni, BT Purwanto, T Widiandani… - Borneo Journal of …, 2024 - journal.umpr.ac.id
Breast cancer remains a significant public health concern, necessitating the discovery of
novel therapeutic agents. This study investigates the potential of thiourea derivatives …
novel therapeutic agents. This study investigates the potential of thiourea derivatives …
4-Methoxyphenethyl (E)-3-(o-tolyl)acrylate
M Santoso, E Pamela, EY Ramadhani, YA Ilfahmi… - Molbank, 2022 - mdpi.com
4-Methoxyphenethyl (E)-3-(o-tolyl) acrylate (1) was obtained in a good yield by the reaction
of 2-methylcinnamic acid, 4-methoxyphenethyl alcohol, 2-methyl-6-nitrobenzoic anhydride …
of 2-methylcinnamic acid, 4-methoxyphenethyl alcohol, 2-methyl-6-nitrobenzoic anhydride …
Investigating Methyl And Nitro Substituents Affect In Para Position On N-Benzoyl-N'-Phenylthiourea Compounds As Potential Treatments For Breast Cancer
D Kesuma, RR Risthanti… - RASĀYAN Journal of …, 2023 - repository.ubaya.ac.id
The primary challenge in chemotherapy for breast cancer stems from the limited
effectiveness of existing drugs due to the diverse mutations, each requiring specific …
effectiveness of existing drugs due to the diverse mutations, each requiring specific …
[PDF][PDF] In-silico ANALYSIS OF (S)-PINOSTROBINBENZOATE DERIVATIVES FROM Boesenbergia pandurata Roxb. AS THE CYCLOOXYGENASE-2 INHIBITORS IN …
ABSTRACT Boesenbergia pandurata Roxb. Schlecht, often known as Temu kunci, contains
the flavonoid pinostrobin in its rhizome. It is useful against inflammation because it can …
the flavonoid pinostrobin in its rhizome. It is useful against inflammation because it can …
[PDF][PDF] MOLECULAR DOCKING OF NOVEL BENZOPYRAN ANALOGUES AND INHIBITION PROPERTIES OF ANTIDIABETIC AGENTS AGAINST α-AMYLASE AND α …
D Bharathi, P Valentina… - Rasayan Journal of …, 2022 - rasayanjournal.co.in
Alpha amylase and alpha-glucosidase inhibitors play a key role in treating diabetes mellitus.
Based on this idea the present study aimed in designing different benzopyran analogs and …
Based on this idea the present study aimed in designing different benzopyran analogs and …