C3‐Functionalization of Imidazo[1,2‐a]pyridines

Z Tashrifi… - European Journal of …, 2020 - Wiley Online Library
Among nitrogen‐containing organic compounds, imidazo [1, 2‐a] pyridines, and especially
C3‐functionalized imidazo [1, 2‐a] pyridines, have a wide range of industrial applications in …

The application of microwaves, ultrasounds, and their combination in the synthesis of nitrogen-containing bicyclic heterocycles

F Frecentese, F Sodano, A Corvino… - International journal of …, 2023 - mdpi.com
The use of alternative energy sources, such as microwaves (MW) or ultrasounds (US), and
their mutual cross-combination have been widely described in the literature in the …

Design, green synthesis, and quorum sensing quenching potential of novel 2-oxo-pyridines containing a thiophene/furan scaffold and targeting a Las R gene on P …

YA Ammar, A Ragab, MA Migahed, S Al-Sharbasy… - RSC …, 2023 - pubs.rsc.org
The current trend in fighting bacteria is attacking the virulence and quorum-sensing (QS)
signals that control bacterial communication and virulence factors, especially biofilm …

One‐Pot Construction of Bis‐Heterocycles through Isocyanide Based Multicomponent Reactions

S Ishwar Bhat - ChemistrySelect, 2020 - Wiley Online Library
Bis‐heterocycles (BHCs) are hybrid molecules comprising two linked, bound, spacer, or
fused heterocyclic skeletons. In recent years, these compounds have attracted increased …

First biocatalytic Groebke-Blackburn-Bienaymé reaction to synthesize imidazo [1, 2-a] pyridine derivatives using lipase enzyme

M Budhiraja, R Kondabala, A Ali, V Tyagi - Tetrahedron, 2020 - Elsevier
In this study, first biocatalytic synthesis of clinically important imidazo [1, 2-a] pyridine based
compounds has been achieved. The Candida antarctica lipase B (CALB) enzyme was found …

Solvent- and Catalyst-Free One-Pot Green Bound-Type Fused Bis-Heterocycles Synthesis via Groebke–Blackburn–Bienaymé Reaction/SNAr/Ring-Chain Azido …

MA Claudio-Catalán, SG Pharande… - ACS …, 2018 - ACS Publications
A new, efficient, green, endogenous water-triggered, solvent-and catalyst-free ultrasound-
assisted one-pot Groebke–Blackburn–Bienaymé reaction/SNAr/ring-chain azido …

Diaza-1, 3-butadienes as useful intermediate in heterocycles synthesis

J Heredia-Moya, DA Zurita, JE Cadena-Cruz… - Molecules, 2022 - mdpi.com
Many heterocyclic compounds can be synthetized using diaza-1, 3-butadienes (DADs) as
key structural precursors. Isolated and in situ diaza-1, 3-butadienes, produced from their …

Ultrasound-assisted synthesis of nitrogen and oxygen containing heterocycles

SK Wahan, G Bhargava… - Current Organic Chemistry, 2023 - benthamdirect.com
Ultrasound is well explored in the preparation of several heterocycles as it is an eco-friendly,
safer and cheaper technique compared to the previous conventional synthetic approach …

Multicomponent one-pot synthesis of luminescent imidazo [1, 2-a] pyridine-3-amines. Studies of fluorescence, solvatochromism, TD-DFT calculations and bioimaging …

M Kurva, MÁ Claudio-Catalán… - Journal of Molecular …, 2023 - Elsevier
Herein we report on a novel series (4a-4p) of fluorescent Imidazo [1, 2-a] pyridines (IMPs)
synthesized via an eco-friendly microwave-assisted Groebke-Blackburn-Bienaymé reaction …

Mechanochemical IMCR and IMCR-post transformation domino strategies: towards the sustainable DOS of dipeptide-like and heterocyclic peptidomimetics

SG Pharande, MA Rentería-Gómez… - New Journal of …, 2022 - pubs.rsc.org
A facile mechanochemical Ugi four-component reaction (MC-Ugi-4CR) has been developed
for the synthesis of new dipeptide-like products in high yields under solvent-, catalyst …