Particular success has been achieved in the synthesis of new products and in processes
since the twelve principles of “green chemistry” were formulated in the 1990s. These …

The synthesis of N-heterocycles is one of the most active areas due to their structures with
extensive applications in the fields of organic, pharmaceutical and materials chemistry. It is …

The unprecedented title reaction between glycine derivatives and indoles, as well as the
auto‐oxidative Povarov/aromatization tandem reaction of glycine derivatives with olefins are …

The Cu/N-ligand/TEMPO catalytic system was first applied to the aerobic oxidative synthesis
of heterocycles. As demonstrated, 2-substituted quinazolines and 4 H-3, 1-benzoxazines …

An efficient Cu-catalyzed synthesis of quinazolines via the C–N bond formation reactions
between N–H bonds of amidines and C (sp3)–H bonds adjacent to sulfur or nitrogen atoms …

Multi-target drugs against selective multiple targets improve therapeutic efficacy, safety and
resistance profiles by collective regulations of a primary therapeutic target together with …

We have developed a visible light-induced photo-redox copper-catalyzed oxidative Csp2–H
annulation (Friedel–Crafts-type cyclization) of amidines with terminal alkynes at room …

A straightforward iron-catalyzed divergent oxidative tandem synthesis of
dihydroquinazolines and quinolines from N-alkylanilines using a TEMPO oxoammonium salt …

A novel and efficient aerobic protocol for the oxidative synthesis of 2-aryl
quinazolinesviabenzyl CH bond amination by a one-pot reaction of arylmethanamines with …

In this paper, we developed a rhodium-catalyzed annulation of vinylene carbonate with
amidines, leading to 4-methylquinazolines with moderate to excellent yields. This procedure …