[PDF][PDF] A review on Pyrazole derivatives of pharmacological potential

A Jamwal, A Javed, V Bhardwaj - J. Pharm. BioSci, 2013 - speronline.com
Pyrazole is five membered heterocyclic rings which is versatile lead compound for designing
potent bioactive agent. The interesting groups of this compound has diverse biological …

Thiazole, thio and semicarbazone derivatives against tropical infective diseases: Chagas disease, human African trypanosomiasis (HAT), leishmaniasis, and malaria

CB Scarim, DH Jornada, MGM Machado… - European journal of …, 2019 - Elsevier
Thiazole, thiosemicarbazone and semicarbazone moieties are privileged scaffolds (acting
as primary pharmacophores) in many compounds that are useful to treat several diseases …

Synthesis, biological screening and in silico studies of new N-phenyl-4-(1, 3-diaryl-1H-pyrazol-4-yl) thiazol-2-amine derivatives as potential antifungal and …

Y Nandurkar, MR Bhoye, D Maliwal… - European Journal of …, 2023 - Elsevier
A new series of N-aryl-4-(1, 3-diaryl-1H-pyrazol-4-yl) thiazol-2-amine,(8a-x) have been
synthesized by a cyclo-condensation reaction of 2-bromo-1-(1, 3-diphenyl-1H-pyrazol-4-yl) …

Synthesis and Biological Screening of New 2-(5-Aryl-1-phenyl-1H-pyrazol-3-yl)-4-aryl Thiazole Derivatives as Potential Antimicrobial Agents

Y Nandurkar, A Shinde, MR Bhoye, S Jagadale… - ACS …, 2023 - ACS Publications
A new series of 2-(5-aryl-1-phenyl-1 H-pyrazol-3-yl)-4-aryl thiazoles (10a–ab) have been
synthesized by a cyclocondensation reaction of 5-aryl-1-phenyl-1 H-pyrazole-3 …

Synthesis, DNA-binding, molecular docking, and cytotoxic activity of a new 4-amino-N-(5-selenocyanatothiazol-2-yl) benzenesulfonamide

ZO Owidah, RM Alansari, MA Gouda… - Journal of Molecular …, 2023 - Elsevier
Abstract Triselenium dicyanide (TSD, 2) was combined with 4-amino-N-(thiazol-2-yl)
benzenesulfonamide (3) in DMSO to form 4-amino-N-(5-selenocyanatothiazol-2-yl) …

Thiadiazole and Thiazole Derivatives as Potential Antimicrobial Agents

Ц Khamitova, D Berillo, A Lozynskyi… - Mini Reviews in …, 2024 - ingentaconnect.com
Background: This review summarizes data on heterocyclic systems with thiadiazole and
thiazole fragments in molecules as promising antimicrobial agents. Introduction: Thiadiazole …

Thiazole compounds with activity against Cryptococcus gattii and Cryptococcus neoformans in vitro

NP de Sá, CI Lino, NC Fonseca, BM Borelli… - European Journal of …, 2015 - Elsevier
Human cryptococcosis can occur as a primary or opportunistic infection and develop as an
acute, subacute, or chronic, systemic infection involving different host organs. We evaluated …

Heterocycle thiazole compounds exhibit antifungal activity through increase in the production of reactive oxygen species in the Cryptococcus neoformans …

NP Sá, CM Lima, CI Lino, PJS Barbeira… - Antimicrobial agents …, 2017 - Am Soc Microbiol
Human cryptococcosis can occur as a primary or opportunistic infection and develops as an
acute, subacute, or chronic systemic infection involving different organs of the host. Given …

Deep eutectic solvent mediated one-pot synthesis of hydrazinyl-4-phenyl-1, 3-thiazoles

M Foroughi Kaldareh, M Mokhtary… - Polycyclic Aromatic …, 2021 - Taylor & Francis
One-pot synthesis of hydrazinyl-4-phenyl-1, 3-thiazole derivatives was developed by three-
component reaction of various ketones or aldehydes, phenacyl chloride, and …

[HTML][HTML] Synthesis and cytotoxicity evaluation of thiosemicarbazones and their thiazole derivatives

SFP Braga, NC Fonseca, JP Ramos… - Brazilian Journal of …, 2016 - SciELO Brasil
The aims of this study were to synthesize a series of thiosemicarbazones and their thiazole
derivatives, to investigate their cytotoxic activity against three human cancers and normal …